SCHEMBL8136268

SCHEMBL8136268

CCc1cc2c(cc1N1CCN(C)CC1)N(C(C)=O)CC2

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 7/20 0.48
TSHR P16473 2/20 0.47
CYP11B2 P19099 3/20 0.46
ALDH1A1 P00352 4/20 0.43
KDM4E B2RXH2 3/20 0.43
HPGD P15428 3/20 0.43
MAPT P10636 2/20 0.42
PKM P14618 1/20 0.42
RECQL P46063 1/20 0.41
HTR1A P08908 3/20 0.41
HTR1D P28221 2/20 0.41
HTR1B P28222 2/20 0.41
DRD2 P14416 1/20 0.40
DRD4 P21917 1/20 0.40
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
DRD3 P35462 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6607580 0.83 HTR1B (0.47) NOTUMCYP11B2ALDH1A1HPGDHTR1A
SCHEMBL6607581 0.83 HTR1B (0.47) NOTUMCYP11B2ALDH1A1HPGDHTR1A
SCHEMBL8155948 0.83 NOTUM (0.54) NOTUMTSHRCYP11B2ALDH1A1KDM4E
SCHEMBL8118270 0.82 NOTUM (0.55) NOTUMTSHRCYP11B2ALDH1A1KDM4E
SCHEMBL8129693 0.82 SLC2A1 (0.49) NOTUMTSHRCYP11B2ALDH1A1KDM4E
SCHEMBL8130919 0.78 NOTUM (0.54) NOTUMTSHRCYP11B2ALDH1A1KDM4E
SCHEMBL8130057 0.78 TSHR (0.46) NOTUMTSHRCYP11B2ALDH1A1KDM4E
SCHEMBL8133031 0.74 NOTUM (0.60) NOTUMTSHRALDH1A1KDM4EMAPT
SCHEMBL7067785 0.74 TSHR (0.52) NOTUMTSHRALDH1A1KDM4EHPGD
SCHEMBL10289633 0.71 NOTUM (0.63) NOTUMTSHRCYP11B2ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1260781-A Indole derivatives having combined 5HT1A, 5HT1B and 5HT1D receptor antagonist activity SMITHKLINE BEECHAM PLC (GB) 2000-07-19 CN disclosed
EP-0975593-A1 INDOLE DERIVATIVES HAVING COMBINED 5HT1A, 5HT1B AND 5HT1D RECEPTOR ANTAGONIST ACTIVITY SMITHKLINE BEECHAM PLC (GB) 2000-02-02 EP disclosed
WO-1998050358-A1 INDOLE DERIVATIVES HAVING COMBINED 5HT1A, 5HT1B AND 5HT1D RECEPTOR ANTAGONIST ACTIVITY SMITHKLINE BEECHAM PLC (GB) 1998-11-12 WO disclosed