SCHEMBL8136394

SCHEMBL8136394

CC1CC2NC(=O)C=C[C@]2(C)[C@@H]2CC[C@]3(C)CC(Oc4ccncc4)C[C@H]3[C@H]12

nearest known ligand 0.45

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
SRD5A1 P18405 12/20 0.45
SRD5A2 P31213 7/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8136389 1.00 SRD5A1 (0.45) SRD5A1SRD5A2
SCHEMBL916376 0.91 SRD5A1 (0.49) SRD5A1SRD5A2
SCHEMBL917557 0.90 SRD5A1 (0.46) SRD5A1SRD5A2
SCHEMBL8139828 0.90 SRD5A1 (0.45) SRD5A1SRD5A2
SCHEMBL8139829 0.90 SRD5A1 (0.45) SRD5A1SRD5A2
SCHEMBL916826 0.89 SRD5A1 (0.45) SRD5A1SRD5A2
SCHEMBL8132557 0.87 SRD5A1 (0.44) SRD5A1SRD5A2
SCHEMBL8132563 0.87 SRD5A1 (0.44) SRD5A1SRD5A2
SCHEMBL8139825 0.86 SRD5A1 (0.46) SRD5A1SRD5A2
SCHEMBL8139822 0.86 SRD5A1 (0.46) SRD5A1SRD5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6143887-A REACTING A 16-METHYLSULFONATE-4-AZA-ANDROSTANONES WITH HYDROXY SUBSTITUTED AROMATIC OR HETEROAROMATIC COMPOUND AND CESIUM CARBONATE IN PRESENCE OF A POLAR APROTIC SOLVENT MERCK & CO., INC. (US) 2000-11-07 US disclosed
WO-1999058551-A1 PROCESS FOR THE STEREOSELECTIVE SYNTHESIS OF 16-SUBSTITUTED-4-AZA-ANDROSTANONES MERCK & CO., INC. (US) 1999-11-18 WO disclosed