SCHEMBL8136830

SCHEMBL8136830

O[C@@H]1C[C@H]2CN(C3=Nc4cc(Cl)ccc4Oc4ccccc43)CCN2C1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 10/20 0.62
DRD4 P21917 6/20 0.62
DRD2 P14416 3/20 0.62
HTR2A P28223 6/20 0.53
ADRA2A P08913 5/20 0.53
HTR1A P08908 5/20 0.53
HTR2C P28335 5/20 0.53
HRH2 P25021 3/20 0.53
HRH1 P35367 3/20 0.53
ADRB2 P07550 2/20 0.53
CHRM2 P08172 2/20 0.53
CHRM4 P08173 2/20 0.53
CHRM5 P08912 2/20 0.53
ADORA3 P0DMS8 2/20 0.53
CHRM1 P11229 2/20 0.53
ADRA2B P18089 2/20 0.53
ADRA2C P18825 2/20 0.53
CHRM3 P20309 2/20 0.53
DRD1 P21728 2/20 0.53
DRD5 P21918 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8136832 1.00 HRH4 (0.62) HRH4DRD4DRD2HTR2AADRA2A
SCHEMBL8119355 1.00 HRH4 (0.62) HRH4DRD4DRD2HTR2AADRA2A
SCHEMBL8121764 1.00 HRH4 (0.62) HRH4DRD4DRD2HTR2AADRA2A
SCHEMBL8137133 1.00 HRH4 (0.62) HRH4DRD4DRD2HTR2AADRA2A
SCHEMBL8121766 1.00 HRH4 (0.62) HRH4DRD4DRD2HTR2AADRA2A
SCHEMBL8134381 0.85 HRH4 (0.61) HRH4DRD4DRD2HTR2AADRA2A
SCHEMBL8134379 0.85 HRH4 (0.61) HRH4DRD4DRD2HTR2AADRA2A
SCHEMBL8135555 0.85 HRH4 (0.56) HRH4DRD4DRD2HTR2AADRA2A
SCHEMBL8135557 0.85 HRH4 (0.56) HRH4DRD4DRD2HTR2AADRA2A
SCHEMBL8126145 0.84 HRH4 (0.63) HRH4DRD4DRD2HTR2AADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0797577-B1 BICYCLIC NONANE AND DECANE COMPOUNDS HAVING DOPAMINE RECEPTOR AFFINITY ALLELIX BIOPHARMA (CA) 2000-07-26 EP disclosed
EP-0797577-A1 BICYCLIC NONANE AND DECANE COMPOUNDS HAVING DOPAMINE RECEPTOR AFFINITY Allelix Biopharmaceuticals Inc. (CA) 1997-10-01 EP disclosed
WO-1996018630-A1 BICYCLIC NONANE AND DECANE COMPOUNDS HAVING DOPAMINE RECEPTOR AFFINITY ALLELIX BIOPHARMACEUTICALS INC. (CA) 1996-06-20 WO disclosed