SCHEMBL8138265

SCHEMBL8138265

Cc1cc2cc(Nc3ccnc4cc(-c5ccc(CNC(C)C)cc5)sc34)ccc2[nH]1

nearest known ligand 0.76

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
EGFR P00533 20/20 0.76
FLT1 P17948 20/20 0.76
KDR P35968 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7126427 0.91 EGFR (0.78) EGFRFLT1KDR
SCHEMBL7117692 0.88 EGFR (0.74) EGFRFLT1KDR
SCHEMBL7117826 0.86 EGFR (0.84) EGFRFLT1KDR
SCHEMBL7126213 0.86 EGFR (1.00) EGFRFLT1KDR
SCHEMBL7127085 0.86 EGFR (0.85) EGFRFLT1KDR
SCHEMBL7123659 0.86 EGFR (0.81) EGFRFLT1KDR
SCHEMBL7115515 0.85 EGFR (0.79) EGFRFLT1KDR
SCHEMBL7118436 0.85 EGFR (0.97) EGFRFLT1KDR
SCHEMBL7124416 0.85 EGFR (0.82) EGFRFLT1KDR
SCHEMBL7123514 0.85 EGFR (1.00) EGFRFLT1KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1028964-A1 THIENOPYRIMIDINE AND THIENOPYRIDINE DERIVATIVES USEFUL AS ANTICANCER AGENTS Pfizer Products Inc. (US) 2000-08-23 EP claimed
WO-1999024440-A1 THIENOPYRIMIDINE AND THIENOPYRIDINE DERIVATIVES USEFUL AS ANTICANCER AGENTS PFIZER PRODUCTS INC. (US) 1999-05-20 WO claimed
EP-1028964-A1 THIENOPYRIMIDINE AND THIENOPYRIDINE DERIVATIVES USEFUL AS ANTICANCER AGENTS Pfizer Products Inc. (US) 2000-08-23 EP disclosed
WO-1999024440-A1 THIENOPYRIMIDINE AND THIENOPYRIDINE DERIVATIVES USEFUL AS ANTICANCER AGENTS PFIZER PRODUCTS INC. (US) 1999-05-20 WO disclosed