SCHEMBL813890

SCHEMBL813890

NC(=O)C1CCC(C(N)=O)C1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.42
MAPT P10636 1/20 0.42
KMT2A Q03164 1/20 0.42
ATM Q13315 1/20 0.42
CYP2D6 P10635 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
NOS2 P35228 1/20 0.40
GAA P10253 1/20 0.35
EPHX1 P07099 2/20 0.35
PLG P00747 1/20 0.35
PLAT P00750 1/20 0.35
LMNA P02545 1/20 0.35
ACE P12821 1/20 0.34
CHRNB2 P17787 3/20 0.33
CHRNA3 P32297 3/20 0.33
CHRNA4 P43681 3/20 0.33
CHRNB4 P30926 2/20 0.33
CHRNA7 P36544 1/20 0.33
GLI1 P08151 1/20 0.32
CHRNB3 Q05901 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15542332 1.00 KDM4E (0.42) KDM4EMAPTKMT2AATMCYP2D6
SCHEMBL31022855 0.97 KDM4E (0.41) KDM4EMAPTKMT2AATMCYP2D6
SCHEMBL31243354 0.89 ACE (0.48) KDM4EMAPTKMT2AATMCYP2D6
SCHEMBL31243364 0.89 ACE (0.48) KDM4EMAPTKMT2AATMCYP2D6
SCHEMBL2401050 0.89 ACE (0.48) KDM4EMAPTKMT2AATMCYP2D6
SCHEMBL24906949 0.89 ACE (0.48) KDM4EMAPTKMT2AATMCYP2D6
SCHEMBL10891462 0.88 KMT2A (0.50) KDM4EMAPTKMT2AATMCYP2D6
SCHEMBL14738046 0.88 KMT2A (0.50) KDM4EMAPTKMT2AATMCYP2D6
SCHEMBL15139869 0.88 KMT2A (0.50) KDM4EMAPTKMT2AATMCYP2D6
SCHEMBL28025415 0.88 KMT2A (0.50) KDM4EMAPTKMT2AATMCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3526261-A1 BETA-NUCLEATED PROPYLENE TERPOLYMER COMPOSITION WITH GOOD TOUGHNESS Borealis AG (AT) 2019-08-21 EP disclosed
WO-2018069263-A1 BETA-NUCLEATED PROPYLENE TERPOLYMER COMPOSITION WITH GOOD TOUGHNESS BOREALIS AG (AT) 2018-04-19 WO disclosed
EP-2350147-A1 PROPYLENE-BUTENE RANDOM COPOLYMER PRODUCED IN THE PRESENCE OF A METTALOCENE CATALYST Borealis AG (AT) 2011-08-03 EP disclosed
EP-2344585-A1 NEW SEWAGE PIPE MATERIAL WITH IMPROVED PROPERTIES Borealis AG (AT) 2011-07-20 EP disclosed
EP-2279216-A1 PROPYLENE-HEXENE RANDOM COPOLYMER PRODUCED IN THE PRESENCE OF A ZIEGLER NATTA CATALYST Borealis AG (AT) 2011-02-02 EP disclosed
WO-2010057841-A1 PROPYLENE-BUTENE RANDOM COPOLYMER PRODUCED IN THE PRESENCE OF A METTALOCENE CATALYST BOREALIS AG (AT) 2010-05-27 WO disclosed
WO-2010057840-A1 PROPYLENE-HEXENE RANDOM COPOLYMER PRODUCED IN THE PRESENCE OF A METALLOCENE CATALYST BOREALIS AG (AT) 2010-05-27 WO disclosed
WO-2010037747-A1 NEW SEWAGE PIPE MATERIAL WITH IMPROVED PROPERTIES BOREALIS AG (AT) 2010-04-08 WO disclosed
WO-2009144166-A1 PROPYLENE-HEXENE RANDOM COPOLYMER PRODUCED IN THE PRESENCE OF A ZIEGLER NATTA CATALYST BOREALIS AG (AT) 2009-12-03 WO disclosed
EP-1495072-A1 SYNTACTIC POLYOLEFIN COMPOSITION FOR PIPE COATING Borealis Technology Oy (FI) 2005-01-12 EP disclosed
WO-2003087205-A1 SYNTACTIC POLYOLEFIN COMPOSITION FOR PIPE COATING BOREALIS TECHNOLOGY OY (FI) 2003-10-23 WO disclosed
WO-1996000729-A2 PROCESS FOR THE PREPARATION OF AZANORADAMANTANE BENZAMIDES G.D. SEARLE & CO. (US) 1996-01-11 WO disclosed