SCHEMBL8142123

SCHEMBL8142123

CC(C)(C)[Si](OC1CC(O)CC(O[Si](c2ccccc2)(c2ccccc2)C(C)(C)C)C1)(c1ccccc1)c1ccccc1

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.35
CYP3A4 P08684 1/20 0.30
HTT P42858 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
SMYD2 Q9NRG4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10549270 1.00 BACE1 (0.35) BACE1CYP3A4HTTSMN1; SMN2SMYD2
SCHEMBL22283784 0.98 BACE1 (0.36) BACE1CYP3A4HTTSMN1; SMN2SMYD2
SCHEMBL870869 0.98 BACE1 (0.36) BACE1CYP3A4HTTSMN1; SMN2SMYD2
SCHEMBL1139920 0.89 BACE1 (0.36) BACE1CYP3A4HTTSMN1; SMN2SMYD2
SCHEMBL1139919 0.89 BACE1 (0.36) BACE1CYP3A4HTTSMN1; SMN2SMYD2
SCHEMBL1560459 0.89 BACE1 (0.36) BACE1CYP3A4HTTSMN1; SMN2SMYD2
SCHEMBL7344125 0.88 BACE1 (0.36) BACE1
SCHEMBL7339050 0.88 BACE1 (0.36) BACE1
SCHEMBL26964687 0.88 BACE1 (0.36) BACE1
SCHEMBL7344545 0.88 BACE1 (0.36) BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4713320-A2 BCAT2 INHIBITORS Agios Pharmaceuticals, Inc. (US) 2026-03-25 EP disclosed
WO-2024238820-A2 BCAT2 INHIBITORS AGIOS PHARMACEUTICALS, INC. (US) 2024-11-21 WO disclosed
EP-4430036-A2 BCAT2 INHIBITORS Agios Pharmaceuticals, Inc. (US) 2024-09-18 EP disclosed
WO-2023086539-A2 BCAT2 INHIBITORS AGIOS PHARMACEUTICALS, INC. (US) 2023-05-19 WO disclosed
US-6013807-A Antitumor tetracyclic compounds UNIVERSITY COLLEGE CARDIFF CONSULTANTS LIMITED (GB) 2000-01-11 US disclosed
US-5852204-A Pyrrolo 3,2-b-!-carbazoles and 1H 1!benzothieno 2,3-f! indoles having anti-tumor activity UNIVERSITY COLLEGE CARDIFF CONSULTANTS LIMITED (GB) 1998-12-22 US disclosed
EP-0741729-A1 ANTITUMOUR TETRACYCLIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1996-11-13 EP disclosed
WO-1995021170-A1 ANTITUMOUR TETRACYCLIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1995-08-10 WO disclosed
US-4841071-A 6-substituted-4-hydroxy-tetrahydropyran-2-ones SANDOZ PHARM. CORP. (US) 1989-06-20 US disclosed
US-4571428-A 6-Substituted-4-hydroxy-tetrahydropyran-2-ones SANDOZ, INC. (US) 1986-02-18 US disclosed