SCHEMBL8143136

SCHEMBL8143136

COC(=O)c1ccc(-c2ccc(N)cc2C(F)(F)F)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.51
GLA P06280 1/20 0.51
POLB P06746 1/20 0.51
TSHR P16473 1/20 0.51
NOTUM Q6P988 2/20 0.50
EGFR P00533 2/20 0.48
MAPT P10636 2/20 0.47
TP53 P04637 1/20 0.47
RAB9A P51151 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
MAPK1 P28482 1/20 0.47
CFTR P13569 3/20 0.44
PDGFRB P09619 1/20 0.44
KDR P35968 1/20 0.44
AKR1C3 P42330 2/20 0.43
AKR1C2 P52895 2/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA9 Q16790 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16255742 0.84 TDP1 (0.53) NOTUMEGFRMAPTRAB9ASMN1; SMN2
SCHEMBL28669018 0.84 SRD5A2 (0.57) POLBTSHRNOTUMEGFRAKR1C3
SCHEMBL497989 0.84 CA12 (0.53) GAANOTUMEGFRTP53AKR1C3
SCHEMBL21300493 0.82 GLA (0.58) GAAGLAPOLBTSHRAKR1C3
SCHEMBL8141484 0.82 GLA (0.58) GAAGLAPOLBTSHRAKR1C3
SCHEMBL12141744 0.82 NOTUM (0.49) POLBNOTUMEGFRAKR1C3AKR1C2
SCHEMBL14791904 0.82 EGFR (0.60) GAANOTUMEGFRAKR1C3AKR1C2
Methoxymethane SCHEMBL28910833 0.82 GLA (0.66) GAAGLAPOLBTSHRAKR1C3
SCHEMBL15920972 0.81 KDM4E (0.55) NOTUMEGFRMAPTSMN1; SMN2AKR1C3
Methyl Alcohol SCHEMBL28910832 0.80 GLA (0.68) GAAGLAPOLBTSHRAKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6100272-A Tetracyclic spiro compounds as 5HT1B receptor antagonists SMITHKLINE BEECHAM P.L.C. (GB) 2000-08-08 US disclosed
EP-0888358-A1 PIPERIDINE DERIVATIVES SMITHKLINE BEECHAM PLC (GB) 1999-01-07 EP disclosed
WO-1997034901-A1 PIPERIDINE DERIVATIVES SMITHKLINE BEECHAM P.L.C. (GB) 1997-09-25 WO disclosed