SCHEMBL8143173

SCHEMBL8143173

CC1[C@@H](C)C[C@@H](C(=O)NCc2cc(Cl)ccc2-n2cnnn2)N1C(=O)C(O)c1ccccc1F

nearest known ligand 0.57

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.57
F2 P00734 13/20 0.55
PRSS1 P07477 2/20 0.55
F9 P00740 1/20 0.55
F10 P00742 1/20 0.55
PLAT P00750 1/20 0.55
F11 P03951 1/20 0.55
KLKB1 P03952 1/20 0.55
F7 P08709 1/20 0.55
TBXA2R P21731 1/20 0.55
PRSS3 P35030 1/20 0.55
KCNH2 Q12809 3/20 0.50
MASP2 O00187 1/20 0.43
F12 P00748 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4211628 0.89 CYP3A4 (0.57) CYP3A4F2PRSS1F9F10
SCHEMBL4206625 0.89 CYP3A4 (0.57) CYP3A4F2PRSS1F9F10
SCHEMBL8144224 0.87 CYP3A4 (0.63) CYP3A4F2PRSS1F9F10
SCHEMBL643641 0.84 CYP3A4 (0.80) CYP3A4F2PRSS1F9F10
SCHEMBL8145574 0.83 CYP3A4 (0.57) CYP3A4F2PRSS1F9F10
SCHEMBL8150553 0.83 CYP3A4 (0.55) CYP3A4F2PRSS1F9F10
SCHEMBL8147627 0.83 F2 (0.56) CYP3A4F2PRSS1F9F10
SCHEMBL641518 0.83 CYP3A4 (0.57) CYP3A4F2PRSS1F9F10
SCHEMBL643295 0.83 CYP3A4 (0.57) CYP3A4F2PRSS1F9F10
SCHEMBL8150385 0.82 F2 (0.54) CYP3A4F2PRSS1F9F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009004383-A2 AZA-BICYCLOHEXANE COMPOUNDS USEFUL AS ANTICOAGULANTS ASTRAZENECA AB (SE) 2009-01-08 WO disclosed