SCHEMBL8145252

SCHEMBL8145252

O=CC(=O)Oc1cc(-c2ccccc2)c(O)c(-c2ccccc2)c1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 5/20 0.50
PTPN1 P18031 4/20 0.45
PTPN6 P29350 2/20 0.43
AKR1C3 P42330 1/20 0.42
AKR1C2 P52895 1/20 0.42
AKR1C1 Q04828 1/20 0.42
EGFR P00533 1/20 0.42
PTPN2 P17706 1/20 0.41
HNF4A P41235 1/20 0.40
HDAC8 Q9BY41 3/20 0.39
HDAC4 P56524 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
PDE4B Q07343 1/20 0.38
HK2 P52789 1/20 0.38
NSD2 O96028 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3273499 0.81 BACE1 (0.75) BACE1PTPN1PDE4B
SCHEMBL8144121 0.77 BACE1 (0.47) BACE1PTPN1PTPN6AKR1C3AKR1C2
SCHEMBL93342 0.75 KMT2A (0.48) NSD2
Water SCHEMBL27382344 0.73 KMT2A (0.47) NSD2
SCHEMBL1706197 0.73 KMT2A (0.47) NSD2
SCHEMBL10711952 0.73 KMT2A (0.47) NSD2
SCHEMBL27509115 0.72 FFAR4 (0.44) BACE1AKR1C3AKR1C2AKR1C1
SCHEMBL9472211 0.72 PTPN1 (0.53) BACE1PTPN1PTPN6AKR1C3AKR1C2
SCHEMBL5989278 0.72 BACE1 (0.73) BACE1HDAC8HDAC4HDAC2PDE4B
SCHEMBL9469340 0.70 PTPN1 (0.63) BACE1PTPN1PTPN6AKR1C3AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6017918-A Phenyl glycine compounds and methods of treating atherosclerosis and restenosis WARNER-LAMBERT COMPANY (US) 2000-01-25 US disclosed