SCHEMBL8148751

SCHEMBL8148751

CCCCCOc1ccc(C(=O)/C=C/c2ccc(OC)c(OC)c2)cc1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.78
KDM4E B2RXH2 2/20 0.78
LMNA P02545 2/20 0.78
TNFRSF1A P19438 2/20 0.71
ABCG2 Q9UNQ0 6/20 0.70
MEN1 O00255 1/20 0.70
KMT2A Q03164 1/20 0.70
CA1 P00915 1/20 0.62
CA2 P00918 1/20 0.62
NPC1 O15118 1/20 0.61
RAB9A P51151 1/20 0.61
ALDH1A1 P00352 1/20 0.61
SMN1; SMN2 Q16637 1/20 0.61
CYP1A1 P04798 1/20 0.59
CYP1A2 P05177 1/20 0.59
CYP2D6 P10635 1/20 0.59
CYP1B1 Q16678 1/20 0.59
DPP4 P27487 1/20 0.59
PTPN1 P18031 1/20 0.59
EGFR P00533 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8148755 1.00 MAPT (0.78) MAPTKDM4ELMNATNFRSF1AABCG2
SCHEMBL9113047 0.93 KDM4E (0.82) MAPTKDM4ELMNATNFRSF1AABCG2
SCHEMBL9113057 0.93 KDM4E (0.82) MAPTKDM4ELMNATNFRSF1AABCG2
SCHEMBL25200497 0.87 MAPT (0.69) MAPTKDM4ELMNATNFRSF1AABCG2
SCHEMBL25209892 0.87 MAPT (0.69) MAPTKDM4ELMNATNFRSF1AABCG2
SCHEMBL29576289 0.87 MAPT (0.76) MAPTKDM4ELMNATNFRSF1AABCG2
SCHEMBL25193831 0.87 MAPT (0.69) MAPTKDM4ELMNATNFRSF1AABCG2
SCHEMBL25218301 0.87 MAPT (0.69) MAPTKDM4ELMNATNFRSF1AABCG2
SCHEMBL30383815 0.87 MAPT (0.69) MAPTKDM4ELMNATNFRSF1AABCG2
SCHEMBL23788887 0.86 ABCG2 (0.84) ABCG2CYP1A1CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0996432-A2 BIOLOGICALLY ACTIVE 1,3-BIS-AROMATIC-PROP-2-EN-1-ONES, 1,3-BIS-AROMATIC-PROPAN-1-ONES, AND 1,3-BIS-AROMATIC-PROP-2-YN-1-ONES STATENS SERUMINSTITUT (DK) 2000-05-03 EP disclosed
WO-1999000114-A2 BIOLOGICALLY ACTIVE 1,3-BIS-AROMATIC-PROP-2-EN-1-ONES, 1,3-BIS-AROMATIC-PROPAN-1-ONES, AND 1,3-BIS-AROMATIC-PROP-2-YN-1-ONES STATENS SERUM INSTITUT (DK) 1999-01-07 WO disclosed