SCHEMBL8148982

SCHEMBL8148982

CC(C)N(C(=O)C1CC[C@H]2[C@@H]3CC=C4C=C(C(=O)O)CC[C@]4(C)[C@@H]3CC[C@]12C)C(C)C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 14/20 1.00
SRD5A1 P18405 2/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8148978 1.00 SRD5A2 (1.00) SRD5A2SRD5A1
SCHEMBL10704713 1.00 SRD5A2 (1.00) SRD5A2SRD5A1
SCHEMBL8158161 0.90 SRD5A2 (0.81) SRD5A2SRD5A1
SCHEMBL8158159 0.90 SRD5A2 (0.81) SRD5A2SRD5A1
SCHEMBL9111609 0.88 SRD5A2 (0.78) SRD5A2SRD5A1
SCHEMBL8802570 0.88 SRD5A2 (0.77) SRD5A2SRD5A1
SCHEMBL8803249 0.88 SRD5A2 (0.77) SRD5A2SRD5A1
SCHEMBL8802666 0.86 SRD5A2 (0.75) SRD5A2SRD5A1
SCHEMBL8149717 0.86 SRD5A2 (0.75) SRD5A2SRD5A1
SCHEMBL8149720 0.86 SRD5A2 (0.75) SRD5A2SRD5A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 25 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0521080-B1 SYNERGISTIC COMPOSITIONS SMITHKLINE BEECHAM CORP (US) 1996-12-11 EP claimed
EP-0684765-A4 TREATING ALOPECIA BY ADMINISTERING 5-ALPHA-REDUCTASE INHIBITING COMPOUNDS. SMITHKLINE BEECHAM CORP (US) 1996-12-04 EP claimed
US-5516768-A Uncompetitive inhibition of steroid and 5α-reductose SMITHKLINE BEECHAM CORPORATION (US) 1996-05-14 US claimed
EP-0684765-A1 TREATING ALOPECIA BY ADMINISTERING 5-ALPHA-REDUCTASE INHIBITING COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1995-12-06 EP claimed
WO-1994017663-A1 TREATING ALOPECIA BY ADMINISTERING 5-ALPHA-REDUCTASE INHIBITING COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1994-08-18 WO claimed
EP-0521080-A4 SYNERGISTIC COMPOSITIONS 1993-11-24 EP claimed
EP-0521080-A1 SYNERGISTIC COMPOSITIONS. SMITHKLINE BEECHAM CORP (US) 1993-01-07 EP claimed
EP-0289327-B1 STEROID 5-ALPHA-REDUCTASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1991-12-18 EP claimed
WO-1991013550-A1 SYNERGISTIC COMPOSITIONS SMITHKLINE BEECHAM CORPORATION (US) 1991-09-19 WO claimed
US-5017568-A Enzyme inhibitors, carboxylation SMITHKLINE BEECHAM CORPORATION (US) 1991-05-21 US claimed
EP-0289327-A2 Steroid 5-alpha-reductase inhibitors SMITHKLINE BEECHAM CORPORATION (US) 1988-11-02 EP claimed
US-6046183-A SYNERGISTIC MIXTURE OF FINASTERIDE AND DOXAZOSIN MERCK & CO., INC. (US) 2000-04-04 US disclosed
US-5994362-A ADMINISTERING FINASTERIDE AND CASODEX MERCK & CO., INC. (US) 1999-11-30 US disclosed
US-5753641-A SYNERGISTIC THERAPY COMPRISING FINASTERIDE AND TERAZOSIN DRUGS MERCK & CO., INC. (US) 1998-05-19 US disclosed
EP-0521080-B1 SYNERGISTIC COMPOSITIONS SMITHKLINE BEECHAM CORP (US) 1996-12-11 EP disclosed
EP-0289327-B1 STEROID 5-ALPHA-REDUCTASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1991-12-18 EP disclosed
WO-1991013550-A1 SYNERGISTIC COMPOSITIONS SMITHKLINE BEECHAM CORPORATION (US) 1991-09-19 WO disclosed
US-5017568-A Enzyme inhibitors, carboxylation SMITHKLINE BEECHAM CORPORATION (US) 1991-05-21 US disclosed
US-4910226-A Estrane compound SMITHKLINE BECKMAN CORPORATION (US) 1990-03-20 US disclosed
EP-0289327-A2 Steroid 5-alpha-reductase inhibitors SMITHKLINE BEECHAM CORPORATION (US) 1988-11-02 EP disclosed