SCHEMBL8155378

SCHEMBL8155378

COc1cc2cc(Br)ccc2cc1C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.46
RXFP1 Q9HBX9 4/20 0.46
NPSR1 Q6W5P4 2/20 0.46
ALDH1A1 P00352 2/20 0.46
PRNP P04156 1/20 0.46
CYP2A6 P11509 1/20 0.43
KDM4E B2RXH2 2/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
POLB P06746 2/20 0.42
MCL1 Q07820 1/20 0.42
NQO2 P16083 4/20 0.41
LMNA P02545 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
THRB P10828 1/20 0.38
NCEH1 Q6PIU2 1/20 0.38
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8147509 1.00 MAPT (0.46) MAPTRXFP1NPSR1ALDH1A1PRNP
SCHEMBL8502354 0.88 CYP2A6 (0.50) MAPTRXFP1NPSR1ALDH1A1PRNP
SCHEMBL8404534 0.81 CYP2A6 (0.56) MAPTALDH1A1CYP2A6KDM4EMEN1
SCHEMBL9381604 0.81 CA12 (0.52) RXFP1PRNPCYP2A6KDM4EMEN1
SCHEMBL17912844 0.80 CYP1A2 (0.54) MAPTALDH1A1CYP2A6KDM4EMEN1
SCHEMBL17912825 0.80 CYP1A2 (0.54) MAPTALDH1A1CYP2A6KDM4EMEN1
SCHEMBL21507510 0.80 CYP2A6 (0.54) MAPTALDH1A1CYP2A6KDM4EMEN1
SCHEMBL15317150 0.80 CYP2A6 (0.54) MAPTALDH1A1CYP2A6KDM4EMEN1
SCHEMBL359387 0.79 POLB (0.52) MAPTNPSR1ALDH1A1CYP2A6KDM4E
SCHEMBL15317151 0.79 PDE4A (0.44) MAPTRXFP1NPSR1ALDH1A1PRNP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040116399-A1 Inhibitors of factor Xa MILLENNIUM PHARMACEUTICALS, INC. 2004-06-17 US disclosed
US-20040116399-A1 Inhibitors of factor Xa MILLENNIUM PHARMACEUTICALS, INC. 2004-06-17 US disclosed