SCHEMBL8156437

SCHEMBL8156437

O=C(O)C(O)(C(=O)c1ccccc1)C(O)(C(=O)O)C(=O)c1ccccc1.O[C@@H]1CCCN[C@@H]1c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.40
CYP2D6 P10635 3/20 0.40
CYP2C19 P33261 2/20 0.40
KDM4E B2RXH2 1/20 0.40
NPC1 O15118 1/20 0.40
HPGD P15428 1/20 0.40
MAPK1 P28482 1/20 0.40
RAB9A P51151 1/20 0.40
TACR1 P25103 4/20 0.39
GBA1 P04062 1/20 0.38
TSHR P16473 3/20 0.36
TP53 P04637 2/20 0.36
CYP3A4 P08684 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
MAPT P10636 1/20 0.36
CYP2C9 P11712 1/20 0.36
THPO P40225 1/20 0.36
HSD17B10 Q99714 1/20 0.36
GMNN O75496 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8108717 0.83 GBA1 (0.52) CYP1A2CYP2D6CYP2C19KDM4ENPC1
SCHEMBL7919080 0.83 GBA1 (0.52) CYP1A2CYP2D6CYP2C19KDM4ENPC1
SCHEMBL6248843 0.83 GBA1 (0.52) CYP1A2CYP2D6CYP2C19KDM4ENPC1
SCHEMBL9205719 0.83 GBA1 (0.52) CYP1A2CYP2D6CYP2C19KDM4ENPC1
SCHEMBL27493818 0.78 TACR1 (0.36) CYP1A2CYP2D6CYP2C19TACR1TSHR
SCHEMBL8156443 0.78 TACR1 (0.36) CYP1A2CYP2D6CYP2C19TACR1TSHR
SCHEMBL8156441 0.76 TP53 (0.54) CYP1A2CYP2D6CYP2C19TACR1GBA1
SCHEMBL8921523 0.75 TACR1 (0.38) TACR1GBA1TSHRMEN1KMT2A
SCHEMBL13966629 0.73 GBA1 (0.55) CYP1A2CYP2D6CYP2C19KDM4ENPC1
SCHEMBL13966630 0.73 GBA1 (0.55) CYP1A2CYP2D6CYP2C19KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6071927-A Spiro-piperidine derivatives and their use as therapeutic agents MERCK SHARP & DOHME LTD. (GB) 2000-06-06 US disclosed