SCHEMBL8165752

SCHEMBL8165752

COC(=O)c1ccc(OC)c2c1OCC(CS)(CS)CO2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.49
ALDH1A1 P00352 6/20 0.49
HSD17B10 Q99714 6/20 0.49
LMNA P02545 3/20 0.49
HPGD P15428 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
GAA P10253 3/20 0.36
KMT2A Q03164 3/20 0.36
MAPT P10636 3/20 0.35
TSHR P16473 2/20 0.35
MAPK1 P28482 2/20 0.35
AGER Q15109 1/20 0.35
CASP1 P29466 1/20 0.34
CASP7 P55210 1/20 0.34
MEN1 O00255 2/20 0.34
POLB P06746 1/20 0.34
HSP90AA1 P07900 1/20 0.33
HTT P42858 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8169222 0.88 KDM4E (0.50) KDM4EALDH1A1HSD17B10LMNAHPGD
SCHEMBL3301916 0.81 KDM4E (0.51) KDM4EALDH1A1HSD17B10LMNAHPGD
SCHEMBL4554858 0.80 KDM4E (0.57) KDM4EALDH1A1HSD17B10LMNAHPGD
SCHEMBL5683830 0.80 KDM4E (0.59) KDM4EALDH1A1HSD17B10LMNASMN1; SMN2
SCHEMBL4467144 0.80 KDM4E (0.73) KDM4EALDH1A1HSD17B10LMNAHPGD
SCHEMBL3307771 0.79 KDM4E (0.49) KDM4EALDH1A1HSD17B10LMNAHPGD
SCHEMBL3302729 0.79 KDM4E (0.49) KDM4EALDH1A1HSD17B10LMNAHPGD
SCHEMBL3302759 0.78 KDM4E (0.51) KDM4EALDH1A1HSD17B10LMNAHPGD
SCHEMBL3305912 0.78 KDM4E (0.51) KDM4EALDH1A1HSD17B10LMNAHPGD
SCHEMBL858141 0.77 KDM4E (0.65) KDM4EALDH1A1HSD17B10LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008104175-A2 NOVEL PHOSPHODIESTERASE INHIBITORS LEO PHARMA A/S (DK) 2008-09-04 WO disclosed