SCHEMBL8167358

SCHEMBL8167358

Cc1nccc(Oc2ccc(-c3ccn(CC4CC4)c(=O)c3N)cc2F)c1C

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 17/20 0.51
BRD4 O60885 2/20 0.38
MET P08581 1/20 0.38
AXL P30530 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2832000 0.86 GRM2 (0.68) GRM2
SCHEMBL8167360 0.83 GRM2 (0.48) GRM2METAXL
SCHEMBL30795030 0.76 GRM2 (0.66) GRM2
SCHEMBL2186047 0.76 GRM2 (0.66) GRM2
SCHEMBL2833898 0.74 GRM2 (0.81) GRM2
SCHEMBL30795860 0.73 GRM2 (0.65) GRM2
SCHEMBL2186805 0.73 GRM2 (0.65) GRM2
SCHEMBL2833971 0.72 GRM2 (0.63) GRM2
SCHEMBL2831898 0.71 GRM2 (0.73) GRM2
SCHEMBL8157229 0.69 GRM2 (0.49) GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008107480-A1 1,4-DISUBSTITUTED 3-CYANO-PYRIDONE DERIVATIVES AND THEIR USE AS POSITIVE MGLUR2 -RECEPTOR MODULATORS ORTHO-MCNEIL-JANSSEN PHARMACEUTICALS, INC (US) 2008-09-12 WO disclosed