SCHEMBL8167479

SCHEMBL8167479

COC(=O)C(=NO)c1ccc(-c2ccccc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.48
MAPT P10636 4/20 0.48
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
CTDSP1 Q9GZU7 1/20 0.46
GAA P10253 1/20 0.46
CYP2C19 P33261 1/20 0.46
LMNA P02545 2/20 0.45
ALDH1A1 P00352 2/20 0.45
EGFR P00533 1/20 0.45
MAPK1 P28482 1/20 0.45
PDCD1 Q15116 1/20 0.45
CD274 Q9NZQ7 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
KDM4E B2RXH2 1/20 0.43
PTPN1 P18031 1/20 0.43
HTT P42858 1/20 0.42
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC1 Q13547 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6025442 0.89 GAA (0.57) SMN1; SMN2MAPTNPC1RAB9AGAA
SCHEMBL6025444 0.89 GAA (0.57) SMN1; SMN2MAPTNPC1RAB9AGAA
SCHEMBL6157370 0.89 GAA (0.57) SMN1; SMN2MAPTNPC1RAB9AGAA
SCHEMBL6191009 0.78 SMN1; SMN2 (0.55) SMN1; SMN2MAPTNPC1RAB9ACTDSP1
Biphenyl SCHEMBL27677322 0.77 TSHR (0.52) SMN1; SMN2MAPTNPC1RAB9ACTDSP1
SCHEMBL8165452 0.76 SMN1; SMN2 (0.43) SMN1; SMN2MAPTNPC1RAB9ALMNA
SCHEMBL8165453 0.76 SMN1; SMN2 (0.43) SMN1; SMN2MAPTNPC1RAB9ALMNA
SCHEMBL19309839 0.75 SMN1; SMN2 (0.52) SMN1; SMN2MAPTNPC1RAB9ACTDSP1
SCHEMBL8894615 0.75 SMN1; SMN2 (0.52) SMN1; SMN2MAPTNPC1RAB9ACTDSP1
SCHEMBL17973397 0.74 SMN1; SMN2 (0.50) SMN1; SMN2MAPTNPC1RAB9ACTDSP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6048852-A BACTERICIDES SMITHKLINE BEECHAM P.L.C. (GB) 2000-04-11 US disclosed
EP-0900197-A1 BETA-THIOPROPIONYL-AMINOACID DERIVATIVES AND THEIR USE AS BETA-LACTAMASE INHIBITORS SMITHKLINE BEECHAM PLC (GB) 1999-03-10 EP disclosed
WO-1997030027-A1 BETA-THIOPROPIONYL-AMINOACID DERIVATIVES AND THEIR USE AS BETA-LACTAMASE INHIBITORS SMITHKLINE BEECHAM PLC (GB) 1997-08-21 WO disclosed