SCHEMBL8167492

SCHEMBL8167492

C=C1c2ccc(C#Cc3ccccc3)cc2CCN1CCN1CCC(O)CC1

nearest known ligand 0.59

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 13/20 0.59
KCNA3 P22001 2/20 0.39
ITGB3 P05106 1/20 0.39
ITGA2B P08514 1/20 0.39
HRH3 Q9Y5N1 3/20 0.39
FFAR1 O14842 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL504310 0.87 GRM5 (0.78) GRM5ITGB3ITGA2BHRH3
SCHEMBL8160743 0.84 HRH3 (0.57) HRH3
SCHEMBL10190619 0.77 GRM5 (0.78) GRM5ITGB3ITGA2BHRH3
SCHEMBL504328 0.74 GRM5 (1.00) GRM5HRH3
SCHEMBL10190617 0.73 GRM5 (0.93) GRM5HRH3
SCHEMBL505037 0.73 GRM5 (0.64) GRM5ITGB3ITGA2BFFAR1
SCHEMBL504287 0.73 GRM5 (1.00) GRM5ITGB3ITGA2BHRH3
SCHEMBL10242676 0.70 HRH3 (0.77) HRH3
SCHEMBL503353 0.68 GRM5 (1.00) GRM5ITGB3ITGA2BHRH3
SCHEMBL504529 0.67 GRM5 (1.00) GRM5ITGB3ITGA2BHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008151184-A1 BENZAMIDE MGLUR5 POSITIVE ALLOSTERIC MODULATORS AND METHODS OF MAKING AND USING SAME VANDERBILT UNIVERSITY (US) 2008-12-11 WO disclosed