SCHEMBL8175233

SCHEMBL8175233

Cc1cc(C)cc(C(=O)N(NC(=O)c2ccccc2)C(C)(C)C)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 6/20 0.82
POLB P06746 1/20 0.77
CYP3A4 P08684 2/20 0.76
CYP2C9 P11712 1/20 0.76

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9511092 0.94 POLB (0.77) ABCB1POLBCYP3A4CYP2C9
SCHEMBL9507281 0.90 CYP3A4 (0.83) ABCB1POLBCYP3A4CYP2C9
SCHEMBL10721518 0.90 ABCB1 (1.00) ABCB1POLBCYP3A4CYP2C9
SCHEMBL5057049 0.90 ABCB1 (0.78) ABCB1POLBCYP3A4CYP2C9
SCHEMBL10721627 0.89 ABCB1 (0.78) ABCB1POLBCYP3A4
Rh-5849 SCHEMBL1538531 0.88 POLB (1.00) ABCB1POLBCYP3A4CYP2C9
SCHEMBL8178344 0.87 ABCB1 (0.84) ABCB1POLBCYP3A4CYP2C9
SCHEMBL10722074 0.87 ABCB1 (0.89) ABCB1POLBCYP3A4CYP2C9
SCHEMBL10718679 0.87 ABCB1 (0.74) ABCB1POLBCYP3A4CYP2C9
SCHEMBL8773665 0.87 POLB (0.85) ABCB1POLBCYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6013836-A PARTICULARLY ACTIVE AGAINST MOTHS AND BEETLES AND THEIR INSECT GROWTH REGULATING ACTIVITY WITHOUT ADVERSE IMPACT ON BENEFICIAL INSECTS; CROPS; FORESTRY ROHM AND HAAS COMPANY (US) 2000-01-11 US disclosed
US-5424333-A Anthelmintic N'-substituted-N,N'-disubstitutedhydrazines ROHM AND HAAS COMPANY (US) 1995-06-13 US disclosed
EP-0361645-B1 ORGANIC HYDRAZINE DERIVATIVES FOR PHARMACEUTICAL USE ROHM AND HAAS COMPANY (US) 1993-09-29 EP disclosed
US-5225443-A Lepidotera and Coleoptera insecticides to protect plants ROHM AND HAAS COMPANY (US) 1993-07-06 US disclosed
EP-0245950-B1 INSECTICIDAL N-SUBSTITUTED-N' - SUBSTITUTED-N, N'-DIACYLHYDRAZINES ROHM AND HAAS COMPANY (US) 1992-06-17 EP disclosed
US-5117057-A Insecticidal N' substituted-N-N'-disubstituted-hydrazines ROHM AND HAAS COMPANY (US) 1992-05-26 US disclosed
EP-0236618-B1 INSECTICIDAL N'-SUBSTITUTED-N,N'-DIACYLHYDRAZINES ROHM AND HAAS COMPANY (US) 1991-02-27 EP disclosed
US-4985461-A Insecticidal N'-substituted-N,N'-diacylhydrazines ROHM AND HAAS COMPANY (US) 1991-01-15 US disclosed
EP-0361645-A2 Organic hydrazine derivatives for pharmaceutical use ROHM AND HAAS COMPANY (US) 1990-04-04 EP disclosed
EP-0245950-A2 Insecticidal n-substituted-n' - substituted-n, n'-diacylhydrazines ROHM AND HAAS COMPANY (US) 1987-11-19 EP disclosed
EP-0236618-A2 Insecticidal N'-substituted-N,N'-diacylhydrazines ROHM AND HAAS COMPANY (US) 1987-09-16 EP disclosed