SCHEMBL8176648

SCHEMBL8176648

CC(C)(C)C(=O)Oc1ccc2c(c1)OC[C@H](c1cccc(C(F)(F)F)c1)[C@@H]2c1ccc(OCCN2CCCC2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 16/20 0.62
ESR2 Q92731 15/20 0.62
CHRM2 P08172 2/20 0.47
ADRA2A P08913 2/20 0.47
ADORA3 P0DMS8 2/20 0.47
CHRM1 P11229 2/20 0.47
SLC6A2 P23975 2/20 0.47
SLC6A4 P31645 2/20 0.47
ADRA1A P35348 2/20 0.47
DRD3 P35462 2/20 0.47
SLC6A3 Q01959 2/20 0.47
KCNH2 Q12809 2/20 0.47
HRH3 Q9Y5N1 2/20 0.47
PGR P06401 1/20 0.47
HTR1A P08908 1/20 0.47
DRD1 P21728 1/20 0.47
TBXA2R P21731 1/20 0.47
PTGS1 P23219 1/20 0.47
OPRM1 P35372 1/20 0.47
HTT P42858 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8176652 1.00 ESR1 (0.62) ESR1ESR2CHRM2ADRA2AADORA3
Hydrochloric Acid SCHEMBL6902006 0.99 ESR1 (0.62) ESR1ESR2CHRM2ADRA2AADORA3
Hydrochloric Acid SCHEMBL8177056 0.99 ESR1 (0.62) ESR1ESR2CHRM2ADRA2AADORA3
Hydrochloric Acid SCHEMBL6902001 0.99 ESR1 (0.62) ESR1ESR2CHRM2ADRA2AADORA3
SCHEMBL6901047 0.93 ESR1 (0.63) ESR1ESR2CHRM2ADRA2AADORA3
SCHEMBL8173012 0.93 ESR1 (0.63) ESR1ESR2CHRM2ADRA2AADORA3
SCHEMBL6901042 0.93 ESR1 (0.63) ESR1ESR2CHRM2ADRA2AADORA3
SCHEMBL8178384 0.89 ESR1 (0.65) ESR1ESR2CHRM2ADRA2AADORA3
SCHEMBL7512960 0.89 ESR1 (0.65) ESR1ESR2CHRM2ADRA2AADORA3
SCHEMBL7512954 0.89 ESR1 (0.65) ESR1ESR2CHRM2ADRA2AADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6043269-A ESTROGEN AGONISTS NOVO NORDISK A/S (DK) 2000-03-28 US disclosed