SCHEMBL8178236

SCHEMBL8178236

C=C1Nc2ccc(F)cc2C2(CCN(CCC(C(=O)N(C)Cc3cccc(F)c3)c3ccc(F)cc3)CC2)O1

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 6/20 0.53
TACR1 P25103 5/20 0.42
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
CCR2 P41597 9/20 0.39
LIPE Q05469 1/20 0.38
CCR5 P51681 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL632868 0.92 TACR3 (0.55) TACR3TACR1MEN1KMT2ACCR2
SCHEMBL632869 0.92 TACR3 (0.55) TACR3TACR1MEN1KMT2ACCR2
SCHEMBL631934 0.87 TACR3 (0.58) TACR3TACR1MEN1KMT2ACCR2
SCHEMBL631631 0.87 TACR3 (0.58) TACR3TACR1MEN1KMT2ACCR2
SCHEMBL631238 0.86 TACR3 (0.62) TACR3TACR1CCR2
SCHEMBL632029 0.85 TACR3 (0.52) TACR3TACR1CCR2CCR5
SCHEMBL632030 0.85 TACR3 (0.52) TACR3TACR1CCR2CCR5
SCHEMBL631383 0.85 TACR3 (0.66) TACR3TACR1MEN1KMT2ACCR2
SCHEMBL631382 0.85 TACR3 (0.66) TACR3TACR1MEN1KMT2ACCR2
SCHEMBL5009009 0.84 TACR3 (0.50) TACR3TACR1CCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008081012-A1 SPIROPIPERIDINE DERIVATIVES AS NK3 ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-07-10 WO disclosed