SCHEMBL8178458

SCHEMBL8178458

O=S(=O)(c1ccccc1)n1cc(-c2cn[nH]c2)c2cc(C3=CCC4(CC3)OCCO4)cnc21

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 5/20 0.37
PTPN11 Q06124 1/20 0.35
HTR6 P50406 8/20 0.35
PDPK1 O15530 1/20 0.33
POLB P06746 1/20 0.33
IKBKE Q14164 1/20 0.33
TBK1 Q9UHD2 1/20 0.33
CCNC P24863 1/20 0.32
CDK8 P49336 1/20 0.32
SUV39H2 Q9H5I1 1/20 0.32
DRD2 P14416 2/20 0.32
HTR2A P28223 2/20 0.32
HTR7 P34969 2/20 0.32
HTR1A P08908 1/20 0.32
CA12 O43570 1/20 0.32
CA9 Q16790 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2753133 0.86 PDPK1 (0.42) BRD4PTPN11HTR6PDPK1POLB
SCHEMBL2752162 0.83 BRD4 (0.36) BRD4PTPN11HTR6PDPK1POLB
SCHEMBL1799609 0.83 BRD4 (0.37) BRD4PTPN11HTR6PDPK1POLB
SCHEMBL2754038 0.83 BRD4 (0.35) BRD4PTPN11HTR6PDPK1POLB
SCHEMBL4555856 0.82 BRD4 (0.36) BRD4PTPN11HTR6PDPK1POLB
SCHEMBL1801618 0.81 BRD4 (0.46) BRD4PTPN11IKBKETBK1SUV39H2
SCHEMBL1801394 0.81 BRD4 (0.35) BRD4PTPN11HTR6POLBIKBKE
SCHEMBL2752379 0.81 PIK3CA (0.45) BRD4PTPN11HTR6IKBKETBK1
SCHEMBL8184787 0.80 POLB (0.36) BRD4PTPN11HTR6POLBCCNC
SCHEMBL8178143 0.78 BRD4 (0.37) BRD4PTPN11HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008095944-A1 7-AZAINDOLE DERIVATIVES AND THEIR USE IN THE INHIBITION OF C-JUN N-TERMINAL KINASE EISAI R&D MANAGEMENT CO. LTD. (JP) 2008-08-14 WO disclosed