SCHEMBL8188564

SCHEMBL8188564

COc1ccc(-c2[nH]nc(-c3ccc(C(N)=O)cc3)c2C)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP10 Q53GL7 2/20 0.55
CA1 P00915 1/20 0.55
CA2 P00918 1/20 0.55
PARP1 P09874 1/20 0.55
PARP2 Q9UGN5 1/20 0.55
PARP4 Q9UKK3 1/20 0.55
MAP4K4 O95819 1/20 0.52
CDK4 P11802 6/20 0.51
CCND1 P24385 6/20 0.51
CCNE2 O96020 5/20 0.51
CCNE1 P24864 5/20 0.51
CDK2 P24941 5/20 0.51
MAPKAPK2 P49137 4/20 0.49
MAP2K4 P45985 2/20 0.49
MAPK1 P28482 1/20 0.49
MAPKAPK3 Q16644 1/20 0.49
MAPK6 Q16659 1/20 0.49
MAPKAPK5 Q8IW41 1/20 0.49
HTT P42858 1/20 0.48
MAPK10 P53779 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2848914 0.81 MAPT (0.55) PARP10CA1CA2PARP1PARP2
SCHEMBL8188562 0.80 CDK2 (0.61) PARP1CDK4CCND1CCNE2CCNE1
SCHEMBL15676819 0.79 MAPT (0.56) PARP10CA1CA2PARP1PARP2
SCHEMBL8185110 0.77 CCNE2 (0.52) CDK4CCND1CCNE2CCNE1CDK2
SCHEMBL5372947 0.76 MAP2K4 (0.66) PARP10CA1CA2PARP1PARP2
SCHEMBL17279998 0.76 CDK4 (0.50) CDK4CCND1CCNE2CCNE1CDK2
SCHEMBL7442028 0.76 PARP10 (0.88) PARP10CA1CA2PARP1PARP2
SCHEMBL27578364 0.75 BACE1 (0.55) PARP10CA1CA2PARP1PARP2
SCHEMBL201761 0.74 PARP10 (1.00) PARP10CA1CA2PARP1PARP2
SCHEMBL1692322 0.73 MAPT (0.53) PARP10CA1CA2PARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000046206-A1 SUBSTITUTED PYRAZOLE BENZYL AMINE DERIVATIVES TO COMBAT ANAEMIAS BAYER AKTIENGESELLSCHAFT (DE) 2000-08-10 WO disclosed