SCHEMBL8192069

SCHEMBL8192069

Cc1cc(C#N)c(C)nc1N

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.46
HSD17B10 Q99714 3/20 0.44
SMN1; SMN2 Q16637 1/20 0.40
ALDH1A1 P00352 6/20 0.39
GAA P10253 2/20 0.39
KHK P50053 1/20 0.39
HTT P42858 2/20 0.38
ADRA2A P08913 1/20 0.38
ADORA2A P29274 1/20 0.38
CSNK1A1 P48729 1/20 0.37
CLK4 Q9HAZ1 1/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
LMNA P02545 2/20 0.35
TSHR P16473 1/20 0.35
HPGD P15428 2/20 0.35
POLB P06746 1/20 0.35
NOS3 P29474 1/20 0.34
NOS1 P29475 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL810713 0.85 KDM4E (0.53) KDM4EHSD17B10SMN1; SMN2ALDH1A1GAA
SCHEMBL16044195 0.84 HTT (0.43) KDM4EHSD17B10SMN1; SMN2ALDH1A1GAA
SCHEMBL19674775 0.80 KDM4E (0.47) KDM4EHSD17B10SMN1; SMN2ALDH1A1GAA
SCHEMBL15537150 0.80 KHK (0.44) KDM4EHSD17B10SMN1; SMN2ALDH1A1GAA
SCHEMBL31214295 0.80 KHK (0.62) KDM4EHSD17B10SMN1; SMN2ALDH1A1GAA
SCHEMBL23860817 0.80 KHK (0.62) KDM4ESMN1; SMN2ALDH1A1GAAKHK
SCHEMBL15568542 0.80 KDM4E (0.42) KDM4EHSD17B10SMN1; SMN2ALDH1A1GAA
SCHEMBL2467905 0.77 KDM4E (0.50) KDM4EHSD17B10SMN1; SMN2ALDH1A1GAA
SCHEMBL2011637 0.77 KDM4E (0.47) KDM4EHSD17B10SMN1; SMN2ALDH1A1GAA
SCHEMBL21604801 0.77 KDM4E (0.41) KDM4EHSD17B10SMN1; SMN2ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6011038-A Pyrazinone thrombin inhibitors MERCK & CO., INC. (US) 2000-01-04 US disclosed