SCHEMBL8199125

SCHEMBL8199125

Cc1c(F)c(N2CCN(C)C(C)C2)cc2c1c(=O)c(C(=O)O)cn2C1CC1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.74
HRH3 Q9Y5N1 1/20 0.74
KDM4E B2RXH2 3/20 0.48
ALDH1A1 P00352 3/20 0.48
LMNA P02545 2/20 0.48
HPGD P15428 2/20 0.48
HSD17B10 Q99714 2/20 0.48
MAPT P10636 1/20 0.48
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
TOP2A P11388 3/20 0.46
TOP2B Q02880 3/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46
CACNA1F O60840 1/20 0.44
POLB P06746 1/20 0.44
MAPK1 P28482 1/20 0.44
CACNA1D Q01668 1/20 0.44
CACNA1S Q13698 1/20 0.44
CACNA1C Q13936 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2738953 0.89 KCNH2 (0.69) KCNH2HRH3KDM4EALDH1A1LMNA
SCHEMBL10109120 0.88 KCNH2 (0.70) KCNH2HRH3KDM4EALDH1A1LMNA
SCHEMBL12665467 0.88 KCNH2 (0.70) KCNH2HRH3KDM4EALDH1A1LMNA
SCHEMBL8556904 0.87 KCNH2 (0.71) KCNH2HRH3KDM4EALDH1A1LMNA
SCHEMBL2738955 0.87 KCNH2 (0.66) KCNH2HRH3KDM4EALDH1A1LMNA
SCHEMBL218555 0.86 KCNH2 (0.65) KCNH2HRH3KDM4EALDH1A1LMNA
SCHEMBL8102436 0.86 KCNH2 (0.70) KCNH2HRH3KDM4EALDH1A1LMNA
Grepafloxacin SCHEMBL29695614 0.85 KCNH2 (1.00) KCNH2HRH3KDM4EALDH1A1LMNA
Grepafloxacin SCHEMBL34157 0.85 KCNH2 (1.00) KCNH2HRH3KDM4EALDH1A1LMNA
Grepafloxacin SCHEMBL34155 0.85 KCNH2 (1.00) KCNH2HRH3KDM4EALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008097546-A2 COMPOUNDS THAT INHIBIT CHOLINESTERASE COLUCID PHARMACEUTICALS, INC. (US) 2008-08-14 WO disclosed