SCHEMBL8199666

SCHEMBL8199666

O=S(=O)(N1CCCN(S(=O)(=O)C(F)(F)F)CCN(S(=O)(=O)C(F)(F)F)CCCN(S(=O)(=O)C(F)(F)F)CC1)C(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.46
KMT2A Q03164 3/20 0.46
POLB P06746 2/20 0.42
GAA P10253 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
ALDH1A1 P00352 3/20 0.37
CA1 P00915 2/20 0.36
CA2 P00918 2/20 0.36
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
HTT P42858 2/20 0.33
PKM P14618 1/20 0.33
CYP17A1 P05093 2/20 0.32
CYP21A2 P08686 2/20 0.32
CYP11B1 P15538 2/20 0.32
GBA1 P04062 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP19A1 P11511 1/20 0.32
SUV39H2 Q9H5I1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3119668 0.97 TSHR (0.42) TSHRKMT2APOLBGAASMN1; SMN2
SCHEMBL1388961 0.92 CA1 (0.43) TSHRKMT2APOLBGAASMN1; SMN2
SCHEMBL7799885 0.92 ESR1 (0.39) TSHRKMT2APOLBSMN1; SMN2CA1
SCHEMBL1319094 0.90 CA1 (0.48) TSHRKMT2APOLBGAASMN1; SMN2
SCHEMBL7856416 0.90 CA1 (0.48) TSHRKMT2APOLBGAASMN1; SMN2
SCHEMBL12225738 0.87 APOBEC3A (0.45) TSHRKMT2APOLBGAAALDH1A1
SCHEMBL799412 0.80 POLB (0.39) TSHRKMT2APOLBSMN1; SMN2L3MBTL1
SCHEMBL31292461 0.80 CA1 (0.34) TSHRKMT2APOLBSMN1; SMN2CA1
SCHEMBL4416229 0.75 ESR1 (0.34) ESR1ESR2CYP17A1CYP21A2CYP11B1
SCHEMBL189725 0.75 KDM4E (0.46) TSHRKMT2AALDH1A1ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6120941-A COMPRISING AN AZA-ETHER BASED COMPOUNDS ACTS AS NEUTRAL RECEPTORS TO COMPLEX THE ANION MOIETY OF THE ELECTROLYTE SALT TO INCREASE THE CONDUCTIVITY IN ALKALI METAL BATTERIES BROOKHAVEN SCIENCE ASSOCIATES (US) 2000-09-19 US disclosed
US-5789585-A IMPROVING CONDUCTIVITY OF ELECTROLYTES IN LITHIUM BATTERIES, COMPLEXING THE ANIONS BROOKHAVEN SCIENCE ASSOCIATES LLC (US) 1998-08-04 US disclosed
US-5705689-A CROWN COMPOUNDS FOR BATTERY ELECTROLYTES WITH LITHIUM IONS ASSOCIATED UNIVERSITIES, INC. (US) 1998-01-06 US disclosed