SCHEMBL8202286

SCHEMBL8202286

Cc1cc(C[C@H]2CN(C)C[C@H]2N)nc(NC(=O)OC(C)(C)C)c1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.36
DYRK1A Q13627 1/20 0.36
SCN9A Q15858 1/20 0.35
LCK P06239 5/20 0.34
TGFBR1 P36897 1/20 0.34
RORC P51449 1/20 0.33
SIRT1 Q96EB6 1/20 0.33
ABL1 P00519 1/20 0.33
SRC P12931 1/20 0.33
BRD4 O60885 2/20 0.32
MAPKAPK2 P49137 1/20 0.32
GRIN2B Q13224 1/20 0.31
SSTR4 P31391 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8209765 1.00 GSK3B (0.36) GSK3BDYRK1ASCN9ALCKTGFBR1
SCHEMBL4727370 0.89 SCN9A (0.36) GSK3BDYRK1ASCN9ALCKTGFBR1
SCHEMBL2257599 0.88 JAK3 (0.35) GSK3BDYRK1ASCN9ALCKBRD4
SCHEMBL2257605 0.88 JAK3 (0.35) GSK3BDYRK1ASCN9ALCKBRD4
SCHEMBL2260109 0.88 JAK3 (0.35) GSK3BDYRK1ASCN9ALCKBRD4
SCHEMBL2261585 0.88 JAK3 (0.35) GSK3BDYRK1ASCN9ALCKBRD4
SCHEMBL2259978 0.88 JAK3 (0.35) GSK3BDYRK1ASCN9ALCKBRD4
SCHEMBL2600843 0.80 SSTR4 (0.35) GSK3BDYRK1ASCN9ALCKSSTR4
SCHEMBL2115673 0.80 SSTR4 (0.35) GSK3BDYRK1ASCN9ALCKSSTR4
SCHEMBL2785572 0.80 SSTR4 (0.35) GSK3BDYRK1ASCN9ALCKSSTR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008042353-A1 POTENT AND HIGHLY SELECTIVE HETEROAROMATIC INHIBITORS OF NEURONAL NITRIC OXIDE SYNTHASE NORTHWESTERN UNIVERSITY (US) 2008-04-10 WO disclosed