SCHEMBL8202872

SCHEMBL8202872

CC(C)[C@@H]1NC(=O)[C@@H](NS(=O)(=O)c2ccc(F)cc2)Cc2ccc(cc2)OCCCCC[C@@H](C(=O)O)NC1=O

nearest known ligand 0.75

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CAPN2 P17655 7/20 0.75
MMP2 P08253 11/20 0.45
MMP7 P09237 11/20 0.45
MMP3 P08254 10/20 0.45
MMP1 P03956 9/20 0.45
CPB2 Q96IY4 1/20 0.42
MMP9 P14780 1/20 0.42
MMP12 P39900 1/20 0.42
MMP13 P45452 1/20 0.42
F2 P00734 1/20 0.39
F10 P00742 1/20 0.39
PLG P00747 1/20 0.39
KLKB1 P03952 1/20 0.39
PROC P04070 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8208871 0.92 CAPN2 (0.74) CAPN2MMP2MMP7MMP3MMP1
SCHEMBL930019 0.89 CAPN2 (0.74) CAPN2MMP2MMP7MMP3MMP1
SCHEMBL8208872 0.86 CAPN2 (1.00) CAPN2MMP2MMP7MMP3MMP1
SCHEMBL930611 0.86 CAPN2 (1.00) CAPN2MMP2MMP7MMP3MMP1
SCHEMBL930382 0.84 CAPN2 (0.76) CAPN2MMP2MMP7MMP3MMP1
SCHEMBL931644 0.83 CAPN2 (1.00) CAPN2MMP2MMP7MMP3MMP1
SCHEMBL931065 0.80 CAPN2 (0.58) CAPN2MMP2MMP7MMP3MMP1
SCHEMBL15869981 0.80 CAPN2 (0.61) CAPN2MMP2MMP7MMP3MMP1
SCHEMBL930579 0.79 CAPN2 (1.00) CAPN2MMP2MMP7MMP3MMP1
SCHEMBL15869976 0.79 CAPN2 (0.59) CAPN2MMP2MMP7MMP3MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008048121-A2 MACROCYCLIC CYSTEINE PROTEASE INHIBITORS AND COMPOSITIONS THEREOF LINCOLN UNIVERSITY (NZ) 2008-04-24 WO disclosed