SCHEMBL8203685

SCHEMBL8203685

CC(C)Oc1cccc(CN2CCC3(CC2)C(=O)N(CCC(=O)O)C(=O)N3c2cccc(F)c2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 11/20 0.44
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
TP53 P04637 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
MAPT P10636 1/20 0.41
ALOX15 P16050 1/20 0.41
TSHR P16473 1/20 0.41
MAPK1 P28482 1/20 0.41
CYP2C19 P33261 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
BACE2 Q9Y5Z0 1/20 0.40
CACNA1F O60840 1/20 0.40
CHRM2 P08172 1/20 0.40
ADRB1 P08588 1/20 0.40
DRD2 P14416 1/20 0.40
SLC6A2 P23975 1/20 0.40
ADRA1D P25100 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3479552 0.88 BACE1 (0.57) BACE1
SCHEMBL8203989 0.82 BACE1 (0.43) BACE1MEN1KMT2ACYP3A4BACE2
SCHEMBL8209469 0.82 BACE1 (0.43) BACE1MEN1KMT2ACACNA1FCHRM2
SCHEMBL8197624 0.80 BACE1 (0.51) BACE1MEN1KMT2ACYP2D6ALOX15
SCHEMBL3479484 0.80 BACE1 (0.56) BACE1
SCHEMBL8269167 0.79 BACE1 (0.49) BACE1MEN1KMT2ACYP2D6ALOX15
SCHEMBL594221 0.79 BACE1 (0.49) BACE1MEN1KMT2ACYP2D6ALOX15
SCHEMBL3479379 0.79 BACE1 (0.59) BACE1
SCHEMBL15146194 0.77 BACE1 (0.45) BACE1MEN1KMT2ACYP2D6ALOX15
SCHEMBL593029 0.77 BACE1 (0.43) BACE1MEN1KMT2ACYP2D6MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008030412-A2 SPIROPIPERIDINE BETA-SECRETASE INHIBITORS FOR THE TREATMENT OF ALZHEIMER'S DISEASE MERCK & CO., INC. (US) 2008-03-13 WO disclosed