SCHEMBL8204916

SCHEMBL8204916

CC(=O)Nc1ccc(CN2CC[C@@]3(C[C@@H]2I)C(=O)NC(=O)N3c2cccc(F)c2)cc1

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 9/20 0.59
BACE2 Q9Y5Z0 1/20 0.59
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
KDM4C Q9H3R0 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
SIGMAR1 Q99720 2/20 0.40
METAP2 P50579 2/20 0.38
POLB P06746 1/20 0.37
MCHR1 Q99705 2/20 0.36
PLD2 O14939 2/20 0.36
PLD1 Q13393 2/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3479450 0.91 BACE1 (0.61) BACE1BACE2KDM4EALDH1A1KDM4C
SCHEMBL3479511 0.77 BACE1 (0.58) BACE1BACE2MCHR1
SCHEMBL3479445 0.77 BACE1 (0.58) BACE1BACE2MCHR1
SCHEMBL3479443 0.77 BACE1 (0.58) BACE1BACE2MCHR1
SCHEMBL2435311 0.76 BACE1 (0.68) BACE1BACE2
SCHEMBL13031126 0.74 BACE1 (0.49) BACE1
SCHEMBL3479612 0.72 BACE1 (0.53) BACE1BACE2KDM4EALDH1A1KDM4C
SCHEMBL592530 0.71 BACE1 (0.60) BACE1BACE2KDM4EALDH1A1KDM4C
SCHEMBL3479509 0.71 BACE1 (0.64) BACE1
SCHEMBL3479463 0.71 BACE1 (0.64) BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008030412-A2 SPIROPIPERIDINE BETA-SECRETASE INHIBITORS FOR THE TREATMENT OF ALZHEIMER'S DISEASE MERCK & CO., INC. (US) 2008-03-13 WO disclosed