SCHEMBL820499

SCHEMBL820499

CO[C@H](C)[C@H](NC(=O)[C@H](C)N(C)C(=O)OC(C)(C)C)C(=O)N1C[C@@H](O)C[C@H]1Cc1c[nH]c2ncccc12

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 2/20 0.33
NTRK1 P04629 2/20 0.32
CYP3A4 P08684 2/20 0.32
CYP2C9 P11712 2/20 0.32
SLC16A1 P53985 2/20 0.32
MTNR1A P48039 1/20 0.31
XIAP P98170 1/20 0.31
BIRC3 Q13489 1/20 0.31
BIRC2 Q13490 1/20 0.31
BIRC7 Q96CA5 1/20 0.31
HTR1A P08908 1/20 0.31
HTR2A P28223 1/20 0.31
HTR7 P34969 1/20 0.31
HTR6 P50406 1/20 0.31
PIK3CD O00329 1/20 0.30
PIK3CA P42336 1/20 0.30
PIK3CB P42338 1/20 0.30
PIK3CG P48736 1/20 0.30
TGM2 P21980 1/20 0.30
MAP2K1 Q02750 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL820181 0.94 NTRK1 (0.35) AURKANTRK1CYP3A4CYP2C9SLC16A1
SCHEMBL818315 0.91 AURKA (0.32) AURKANTRK1MTNR1A
SCHEMBL820497 0.91 AURKA (0.32) AURKANTRK1MTNR1A
SCHEMBL13787025 0.91 AURKA (0.32) AURKANTRK1MTNR1A
SCHEMBL823072 0.85 XIAP (0.43) CYP3A4CYP2C9SLC16A1MTNR1AXIAP
SCHEMBL818633 0.85 XIAP (0.43) CYP3A4CYP2C9SLC16A1MTNR1AXIAP
SCHEMBL13787021 0.80
SCHEMBL820496 0.79 SSTR3 (0.35) CYP3A4MTNR1A
SCHEMBL818314 0.77 HCRTR1 (0.31) MTNR1A
SCHEMBL818000 0.72 XIAP (0.36) AURKANTRK1CYP3A4CYP2C9SLC16A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110288116-A1 IAP INHIBITORS TETRALOGIC PHARMACEUITCAL CORPORATION (US) 2011-11-24 US disclosed
US-20110288116-A1 IAP INHIBITORS TETRALOGIC PHARMACEUITCAL CORPORATION (US) 2011-11-24 US disclosed
WO-2009094287-A1 IAP INHIBITORS TETRALOGIC PHARMACEUTICAL CORPORATION (US) 2009-07-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110288116-A1 IAP INHIBITORS XIAP, BIRC5, BIRC7 AURKA 1959/4885NTRK1 4793/4885CYP3A4 4692/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.