SCHEMBL8205630

SCHEMBL8205630

O=C1NC(=O)c2c1c(CCO)cc1ccccc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 8/20 0.40
CCND1 P24385 8/20 0.40
CCNE2 O96020 4/20 0.40
CCNE1 P24864 4/20 0.40
CDK2 P24941 4/20 0.40
GPR84 Q9NQS5 2/20 0.40
GSK3B P49841 4/20 0.38
DHODH Q02127 1/20 0.38
CDK5 Q00535 3/20 0.37
CDK5R1 Q15078 3/20 0.37
GSK3A P49840 2/20 0.37
CHEK1 O14757 2/20 0.36
WEE1 P30291 1/20 0.36
KMT2A Q03164 3/20 0.36
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
CCNB2 O95067 2/20 0.36
PRKCG P05129 2/20 0.36
PRKCB P05771 2/20 0.36
CDK1 P06493 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9556428 0.81 CDK4 (0.39) CDK4CCND1CCNE2CCNE1CDK2
SCHEMBL15557199 0.80 CDK4 (0.41) CDK4CCND1CCNE2CCNE1CDK2
SCHEMBL4422539 0.78 SLC6A4 (0.47) CDK4CCND1GSK3BCHEK1WEE1
SCHEMBL17045728 0.76 CDK4 (0.37) CDK4CCND1CCNE2CCNE1CDK2
SCHEMBL1756365 0.76 TRPM4 (0.48) CDK4CCND1CCNE2CCNE1CDK2
SCHEMBL8853276 0.76 CDK4 (0.40) CDK4CCND1GPR84GSK3BCDK5
SCHEMBL789452 0.75 TRPM4 (0.47) CDK4CCND1CCNE2CCNE1CDK2
SCHEMBL29128557 0.74 CDK4 (0.39) CDK4CCND1CCNE2CCNE1CDK2
SCHEMBL27814900 0.74 NPC1 (0.55) CDK4CCND1GSK3BDHODHKMT2A
SCHEMBL7767469 0.73 MEN1 (0.50) CDK4GPR84CHEK1WEE1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6096758-A 3-METHYLIMIDAZOPYRIDINES USED FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 2000-08-01 US disclosed