SCHEMBL8206087

SCHEMBL8206087

C=S(=O)(Cc1cc(N2CCOC[C@@H]2C)nc(-c2ccc(N)cc2)n1)c1ccncc1

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 11/20 0.57
PIK3CD O00329 6/20 0.57
MTOR P42345 6/20 0.56
PDCD1 Q15116 10/20 0.55
CD274 Q9NZQ7 10/20 0.55
ATR Q13535 9/20 0.55
CHEK1 O14757 8/20 0.55
ATRIP Q8WXE1 8/20 0.55
ATM Q13315 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3603549 0.91 PIK3CA (0.57) PIK3CAPIK3CDMTORPDCD1CD274
SCHEMBL739897 0.86 PIK3CA (0.72) PIK3CAPIK3CDMTORPDCD1CD274
SCHEMBL3593430 0.84 PIK3CA (0.63) PIK3CAPIK3CDMTORPDCD1CD274
SCHEMBL11924836 0.84 PIK3CA (0.55) PIK3CAPIK3CDMTORPDCD1CD274
SCHEMBL3594878 0.83 PIK3CA (0.61) PIK3CAPIK3CDMTORPDCD1CD274
SCHEMBL13283710 0.83 PIK3CA (0.61) PIK3CAPIK3CDMTORPDCD1CD274
SCHEMBL3605292 0.83 PIK3CA (0.60) PIK3CAPIK3CDMTORPDCD1CD274
SCHEMBL3588785 0.83 PIK3CA (0.60) PIK3CAPIK3CDMTORPDCD1CD274
SCHEMBL3596780 0.83 PIK3CA (0.60) PIK3CAPIK3CDMTORPDCD1CD274
SCHEMBL3602515 0.82 PIK3CA (0.50) PIK3CAPIK3CDMTORPDCD1CD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008023159-A1 MORPHOLINO PYRIMIDINE DERIVATIVES USEFUL IN THE TREATMENT OF PROLIFERATIVE DISORDERS ASTRAZENECA AB (SE) 2008-02-28 WO disclosed