SCHEMBL8207326

SCHEMBL8207326

CC(c1ccccc1)N1C[C@@H](CO)CC1=O

nearest known ligand 0.63

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.63
MAPK1 P28482 1/20 0.51
BRD4 O60885 1/20 0.46
GRM5 P41594 1/20 0.41
HSD11B1 P28845 2/20 0.40
HSD17B2 P37059 1/20 0.39
CYP2D6 P10635 1/20 0.39
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
MAPT P10636 1/20 0.37
P2RX3 P56373 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL576462 1.00 KMT2A (0.63) KMT2AMAPK1BRD4GRM5HSD11B1
SCHEMBL523900 1.00 KMT2A (0.63) KMT2AMAPK1BRD4GRM5HSD11B1
SCHEMBL27902911 1.00 KMT2A (0.63) KMT2AMAPK1BRD4GRM5HSD11B1
SCHEMBL5626616 1.00 KMT2A (0.63) KMT2AMAPK1BRD4GRM5HSD11B1
SCHEMBL576463 1.00 KMT2A (0.63) KMT2AMAPK1BRD4GRM5HSD11B1
SCHEMBL4529849 1.00 KMT2A (0.63) KMT2AMAPK1BRD4GRM5HSD11B1
SCHEMBL523899 1.00 KMT2A (0.63) KMT2AMAPK1BRD4GRM5HSD11B1
SCHEMBL9987097 0.90 KMT2A (0.53) KMT2AMAPK1BRD4GRM5HSD11B1
SCHEMBL14405525 0.89 KMT2A (0.60) KMT2AMAPK1BRD4GRM5HSD11B1
SCHEMBL20306298 0.87 KMT2A (0.48) KMT2AMAPK1BRD4HSD11B1HSD17B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104812753-A Substituted pyridopyrazines as syk inhibitors HUTCHISON MEDIPHARMA LTD 2015-07-29 CN disclosed
CN-101862317-A The pregabalin derivant that is used for the treatment of fibromyalgia and other disease WARNER LAMBERT CO 2010-10-20 CN disclosed
CN-1310872-C Mono- and disubstituted 3-propyl gamma-aminobutyric acids WARNER LAMBERT CO (US) 2007-04-18 CN disclosed
CN-1726023-A Pregabalin derivatives for the treatment of fibromyalgia and other diseases WARNER LAMBERT CO (US) 2006-01-25 CN disclosed
CN-1660779-A Mono- and disubstituted 3-propyl gamma-aminobutyric acids WARNER LAMBERT CO (US) 2005-08-31 CN disclosed
CN-1625393-A Alpha 2 delta ligands to treat tinnitus WARNER LAMBERT CO (US) 2005-06-08 CN disclosed
CN-1196671-C Mono-and disubstituted 3-propyl-gamma-aminobutyric acids WARNER LAMBERT CO (US) 2005-04-13 CN disclosed
CN-1355784-A Mono-and disubstituted 3-propyl-gamma-aminobutyric acids WARNER LAMBERT CO (US) 2002-06-26 CN disclosed
US-6121272-A Bidentate metalloprotease inhibitors THE PROCTER & GAMBLE COMPANY (US) 2000-09-19 US disclosed