SCHEMBL8207401

SCHEMBL8207401

NC1CN(C(=O)OCC(F)(F)F)c2cc(F)c(F)cc2NC1=O

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.36
NR1H2 P55055 1/20 0.32
NR1H3 Q13133 1/20 0.32
FAAH O00519 1/20 0.31
MGLL Q99685 1/20 0.31
ADORA2B P29275 1/20 0.30
IDH1 O75874 1/20 0.30
JAK2 O60674 1/20 0.30
JAK1 P23458 1/20 0.30
JAK3 P52333 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4995341 1.00 HTR2C (0.36) HTR2CNR1H2NR1H3FAAHMGLL
Hydrochloric Acid SCHEMBL4995346 0.99 HTR2C (0.36) HTR2CNR1H2NR1H3FAAHMGLL
Hydrochloric Acid SCHEMBL4995321 0.99 HTR2C (0.36) HTR2CNR1H2NR1H3FAAHMGLL
SCHEMBL4247929 0.83 GAA (0.44)
Hydrochloric Acid SCHEMBL4247932 0.82 GAA (0.43)
Hydrochloric Acid SCHEMBL4247924 0.82 GAA (0.43)
SCHEMBL4993633 0.79 GAA (0.36) HTR2CNR1H2NR1H3
SCHEMBL4993646 0.79 GAA (0.36) HTR2CNR1H2NR1H3
SCHEMBL4992925 0.78 NR1H2 (0.32) NR1H2NR1H3FAAHMGLL
SCHEMBL8209097 0.78 NR1H2 (0.32) NR1H2NR1H3FAAHMGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008034735-A2 4-OXO-2,3,4,5-TETRAHYDRO-BENZO[B][1,4]DIAZEPINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-03-27 WO disclosed