SCHEMBL8207412

SCHEMBL8207412

NC1CN(CCOCc2ccccc2)c2ccccc2N(CC(F)(F)F)C1=O

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 7/20 0.38
PKM P14618 4/20 0.37
DPP4 P27487 1/20 0.36
DPP8 Q6V1X1 1/20 0.36
DPP7 Q9UHL4 1/20 0.36
GAA P10253 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
LTA4H P09960 1/20 0.34
ALDH1A1 P00352 1/20 0.34
AOC3 Q16853 1/20 0.34
SCN10A Q9Y5Y9 1/20 0.34
LIPG Q9Y5X9 1/20 0.33
MAPT P10636 1/20 0.32
ATM Q13315 1/20 0.32
TEAD3 Q99594 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8206826 1.00 SCN9A (0.38) SCN9APKMDPP4DPP8DPP7
Hydrochloric Acid SCHEMBL4994773 0.99 SCN9A (0.38) SCN9APKMDPP4DPP8DPP7
Hydrochloric Acid SCHEMBL4994783 0.99 SCN9A (0.38) SCN9APKMDPP4DPP8DPP7
SCHEMBL8209635 0.92 GAA (0.36) SCN9APKMDPP4DPP8DPP7
Hydrochloric Acid SCHEMBL4993551 0.91 GAA (0.35) SCN9APKMDPP4DPP8DPP7
SCHEMBL4992313 0.79 SCN9A (0.60) SCN9ASCN10A
SCHEMBL4992322 0.79 SCN9A (0.60) SCN9ASCN10A
SCHEMBL14093724 0.76 GAA (0.39) DPP4DPP8DPP7GAAMEN1
SCHEMBL4988616 0.76 GAA (0.39) DPP4DPP8DPP7GAAMEN1
Hydrochloric Acid SCHEMBL4988622 0.75 GAA (0.38) DPP4DPP8DPP7GAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008034735-A2 4-OXO-2,3,4,5-TETRAHYDRO-BENZO[B][1,4]DIAZEPINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-03-27 WO disclosed