SCHEMBL8209547

SCHEMBL8209547

CC(C)Oc1cccc(CN2CC[C@@]3(C[C@@H]2I)C(=O)N(CCNC(=O)c2ccccc2)C(=O)N3c2cccc(N)c2)c1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 1/20 0.37
BACE1 P56817 6/20 0.37
REN P00797 1/20 0.36
CTSD P07339 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
OPRK1 P41145 1/20 0.34
DRD4 P21917 1/20 0.34
CACNA1G O43497 2/20 0.34
SLC5A7 Q9GZV3 1/20 0.34
PLD2 O14939 1/20 0.33
PLD1 Q13393 1/20 0.33
LMNA P02545 1/20 0.33
RECQL P46063 1/20 0.33
GCGR P47871 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3479378 0.85 BACE1 (0.52) BACE1PLD2PLD1
SCHEMBL3479498 0.83 BACE1 (0.41) ENPP2BACE1DRD4
SCHEMBL8203348 0.77 BACE1 (0.45) BACE1OPRM1
SCHEMBL8203688 0.75 BACE1 (0.42) BACE1
SCHEMBL3479552 0.72 BACE1 (0.57) BACE1
SCHEMBL3479379 0.71 BACE1 (0.59) BACE1
SCHEMBL3479484 0.71 BACE1 (0.56) BACE1
SCHEMBL4257463 0.69 BACE1 (0.55) BACE1
SCHEMBL3479588 0.69 BACE1 (0.55) BACE1
SCHEMBL3479586 0.68 BACE1 (0.57) BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008030412-A2 SPIROPIPERIDINE BETA-SECRETASE INHIBITORS FOR THE TREATMENT OF ALZHEIMER'S DISEASE MERCK & CO., INC. (US) 2008-03-13 WO disclosed