SCHEMBL8209729

SCHEMBL8209729

Cc1cc(I)c(Sc2nc3c(N)nccc3n2CCNCCCC(=O)NO)cc1C

nearest known ligand 0.64

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 20/20 0.64
HSP90AB1 P08238 5/20 0.64
HDAC3 O15379 1/20 0.55
HDAC4 P56524 1/20 0.55
HDAC1 Q13547 1/20 0.55
HDAC7 Q8WUI4 1/20 0.55
HDAC2 Q92769 1/20 0.55
HDAC10 Q969S8 1/20 0.55
HDAC11 Q96DB2 1/20 0.55
HDAC8 Q9BY41 1/20 0.55
HDAC6 Q9UBN7 1/20 0.55
HDAC9 Q9UKV0 1/20 0.55
HDAC5 Q9UQL6 1/20 0.55
CDC37 Q16543 1/20 0.54
HSP90B1 P14625 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8151991 0.88 HSP90AA1 (0.68) HSP90AA1HSP90AB1HDAC3HDAC4HDAC1
SCHEMBL8152895 0.87 HSP90AA1 (0.84) HSP90AA1HSP90AB1HDAC3HDAC4HDAC1
SCHEMBL8158943 0.85 HSP90AA1 (0.85) HSP90AA1HSP90AB1HDAC3HDAC4HDAC1
SCHEMBL8204526 0.84 HSP90AA1 (0.87) HSP90AA1HSP90AB1HDAC3HDAC4HDAC1
SCHEMBL8153203 0.84 HSP90AA1 (0.87) HSP90AA1HSP90AB1HDAC3HDAC4HDAC1
SCHEMBL4480998 0.78 HSP90AA1 (1.00) HSP90AA1HSP90AB1HDAC3HDAC4HDAC1
SCHEMBL4900367 0.78 HSP90AA1 (1.00) HSP90AA1HSP90AB1HDAC3HDAC4HDAC1
SCHEMBL8146229 0.74 HSP90AA1 (0.94) HSP90AA1HSP90AB1HDAC3HDAC4HDAC1
SCHEMBL4130807 0.72 HSP90AA1 (1.00) HSP90AA1HSP90AB1CDC37HSP90B1
SCHEMBL8146240 0.71 HSP90AA1 (0.98) HSP90AA1HSP90AB1HDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008033747-A9 MULTI-FUNCTIONAL SMALL MOLECULES AS ANTI-PROLIFERATIVE AGENTS CURIS INC (MA) 2008-07-24 WO disclosed
WO-2008033747-A2 MULTI-FUNCTIONAL SMALL MOLECULES AS ANTI-PROLIFERATIVE AGENTS CURIS, INC. (US) 2008-03-20 WO disclosed