SCHEMBL8209947

SCHEMBL8209947

COCCNCCc1cccc(F)c1

nearest known ligand 0.60

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.60
NOS1 P29475 2/20 0.51
NOS3 P29474 1/20 0.51
KDM4E B2RXH2 2/20 0.50
ALDH1A1 P00352 1/20 0.47
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
HTR2A P28223 2/20 0.46
SCN8A Q9UQD0 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24965971 0.83 TAAR1 (0.57) TAAR1
SCHEMBL12500551 0.81 TAAR1 (0.65) TAAR1NOS1NOS3KDM4EALDH1A1
SCHEMBL10201988 0.81 KDM4E (0.47) KDM4EALDH1A1
SCHEMBL21089609 0.81 TAAR1 (0.60) TAAR1KDM4EALDH1A1MEN1KMT2A
SCHEMBL22566654 0.80 TAAR1 (0.68) TAAR1NOS1NOS3KDM4EMEN1
SCHEMBL14608016 0.80 TAAR1 (0.53) TAAR1SCN8A
SCHEMBL14566080 0.80 TAAR1 (0.55) TAAR1KDM4EALDH1A1KMT2A
SCHEMBL7235032 0.79 GAA (0.65) TAAR1KDM4EMEN1KMT2A
SCHEMBL31114405 0.78 TAAR1 (0.67) TAAR1NOS1NOS3KDM4E
SCHEMBL2257962 0.78 TAAR1 (0.61) TAAR1NOS1NOS3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008042353-A1 POTENT AND HIGHLY SELECTIVE HETEROAROMATIC INHIBITORS OF NEURONAL NITRIC OXIDE SYNTHASE NORTHWESTERN UNIVERSITY (US) 2008-04-10 WO disclosed