SCHEMBL821280

SCHEMBL821280

COC(CCCCCCl)OC

nearest known ligand 0.39

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.39
ALDH1A1 P00352 2/20 0.39
TDP1 Q9NUW8 2/20 0.30
SMPD1 P17405 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11467129 1.00 TSHR (0.39) TSHRALDH1A1TDP1SMPD1
SCHEMBL8053054 0.97 TSHR (0.35) TSHRALDH1A1TDP1
SCHEMBL1769976 0.89
SCHEMBL31543742 0.86 TSHR (0.32) TSHRALDH1A1TDP1
SCHEMBL5160133 0.86 SMPD1 (0.36) SMPD1
SCHEMBL7934687 0.86 SMPD1 (0.36) SMPD1
SCHEMBL7936797 0.86 SMPD1 (0.36) SMPD1
SCHEMBL7934735 0.86 SMPD1 (0.36) SMPD1
SCHEMBL6567377 0.86 SMPD1 (0.36) SMPD1
SCHEMBL6298010 0.83 SMPD1 (0.32) SMPD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 123 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4025246-A2 IMMUNOGENIC COMPOSITIONS AGAINST ENTERIC DISEASES AND METHODS FOR ITS PREPARATION THEREOF Serum Institute Of India Private Limited (IN) 2022-07-13 EP claimed
CN-114728053-A Immunogenic compositions against intestinal disease and process for preparing same 印度血清研究所私人有限公司 2022-07-08 CN claimed
WO-2021044436-A2 IMMUNOGENIC COMPOSITIONS AGAINST ENTERIC DISEASES AND METHODS FOR ITS PREPARATION THEREOF SERUM INSTITUTE OF INDIA PRIVATE LIMITED (IN) 2021-03-11 WO claimed
EP-2387417-B1 BROAD SPECTRUM VACCINE AGAINST NON-TYPHOIDAL SALMONELLA UNIV MARYLAND (US) 2016-05-11 EP claimed
US-9050283-B2 Broad spectrum vaccine against non-typhoidal Salmonella UNIVERSITY OF MARYLAND, BALTIMORE (US) 2015-06-09 US claimed
CN-102964287-B Synthesis method of 3-(4-chlorobutyl)-5-cyanoindole SUZHOU UUGENE BIOPHARMA CO LTD 2014-04-09 CN claimed
CN-102964287-A New synthesis method of 3-(4-chlorobutyl)-5-cyanoindole SUZHOU UUGENE BIOPHARMA CO LTD 2013-03-13 CN claimed
WO-2012061400-A2 METHOD FOR REDUCTION OF FREE POLYSACCHARIDE IN POLYSACCHARIDE-PROTEIN VACCINES REACTIONS USING ION-EXCHANGE MATRICES UNIVERSITY OF MARYLAND, BALTIMORE (US) 2012-05-10 WO claimed
EP-2387417-A2 BROAD SPECTRUM VACCINE AGAINST NON-TYPHOIDAL SALMONELLA University of Maryland, Baltimore (US) 2011-11-23 EP claimed
US-20110274714-A1 Broad Spectrum Vaccine Against Non-Typhoidal Salmonella UNIVERSITY OF MARYLAND, BALTIMORE (US) 2011-11-10 US claimed
US-20040115214-A1 Lipooligosaccharide-based vaccine for prevention of Moraxella (Branhamella) catarrhalis infections in humans GU XIN-XING (US) 2004-06-17 US claimed
US-6685949-B1 OTITIS MEDIA AND SINUSITIS; DETOXIFIED BY TREATING TO REMOVE ESTERIFIED FATTY ACIDS, IMMUNOGENIC CARRIER PROTEIN COVALENTLY LINKED THERETO THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH & HUMAN SERVICES 2004-02-03 US claimed
WO-2003070282-A2 SYNTHESIS OF LIPOPOLYSACCHARIDE-PROTEIN CONJUGATE VACCINES VIA THE LIPID A REGION FOLLOWING REMOVAL OF THE GLYCOSIDIC PHOSPHATE RESIDUE NATIONAL RESEARCH COUNCIL OF CANADA (CA) 2003-08-28 WO claimed
US-6607725-B2 Complex of lipooligosaccharide and immunology carriers THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES 2003-08-19 US claimed
US-6531131-B1 Neisseria meningitidis lipooligosaccharide from which at least one primary O-linked fatty acid has been removed to detoxify it, covalently linked to immunogenic carrier THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES 2003-03-11 US claimed
US-20020001589-A1 Conjugate vaccine for nontypeable haemophilus influenzae GU XIN-XING (US) 2002-01-03 US claimed
US-6207157-B1 OLIGOSACCHARIDE THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES 2001-03-27 US claimed
EP-1047447-A1 LIPOOLIGOSACCHARIDE-BASED VACCINE FOR PREVENTION OF $i(MORAXELLA) $i((BRANHAMELLA)) $i(CATARRHALIS) INFECTIONS IN MAMMALS THE UNITED STATES GOVERNMENT as represented by THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2000-11-02 EP claimed
WO-1999036086-A1 LIPOOLIGOSACCHARIDE-BASED VACCINE FOR PREVENTION OF MORAXELLA (BRANHAMELLA) CATARRHALIS INFECTIONS IN MAMMALS THE GOVERNMENT OF THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1999-07-22 WO claimed
WO-1998026799-A1 CONJUGATE VACCINE FOR SALMONELLA PARATYPHI A THE GOVERNMENT OF THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1998-06-25 WO claimed