SCHEMBL8213995

SCHEMBL8213995

COC(=O)/C=C/c1ccc(OCCCc2ccccc2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B10 O60218 4/20 0.61
AKR1B1 P15121 4/20 0.61
KMT2A Q03164 2/20 0.59
MEN1 O00255 1/20 0.59
ALDH1A1 P00352 1/20 0.59
LMNA P02545 1/20 0.59
S1PR1 P21453 5/20 0.59
S1PR3 Q99500 4/20 0.59
PPARG P37231 2/20 0.58
PPARA Q07869 2/20 0.58
GSK3B P49841 1/20 0.56
BACE1 P56817 1/20 0.56
FFAR1 O14842 1/20 0.55
ALOX5 P09917 1/20 0.54
MAOB P27338 1/20 0.53
PLAAT3 P53816 1/20 0.53
PLAAT5 Q96KN8 1/20 0.53
PLAAT2 Q9NWW9 1/20 0.53
PLAAT4 Q9UL19 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5207328 0.89 PPARA (0.58) KMT2APPARAGSK3BBACE1SMN1; SMN2
SCHEMBL2776601 0.85 GSK3B (0.76) KMT2AMEN1GSK3BBACE1MAOB
SCHEMBL2776603 0.85 GSK3B (0.76) KMT2AMEN1GSK3BBACE1MAOB
SCHEMBL142092 0.83 ABCG2 (0.62) PPARAGSK3BSMN1; SMN2
SCHEMBL8782823 0.83 ABCG2 (0.62) PPARAGSK3BSMN1; SMN2
SCHEMBL451121 0.82 S1PR1 (0.61) AKR1B10AKR1B1KMT2AMEN1ALDH1A1
SCHEMBL451122 0.82 S1PR1 (0.61) AKR1B10AKR1B1KMT2AMEN1ALDH1A1
SCHEMBL9339002 0.82 CA12 (0.57) KMT2ALMNAPPARAGSK3BSMN1; SMN2
SCHEMBL9339004 0.82 CA12 (0.57) KMT2ALMNAPPARAGSK3BSMN1; SMN2
SCHEMBL14634380 0.82 CA12 (0.57) KMT2ALMNAPPARAGSK3BSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008033747-A9 MULTI-FUNCTIONAL SMALL MOLECULES AS ANTI-PROLIFERATIVE AGENTS CURIS INC (MA) 2008-07-24 WO disclosed
WO-2008033747-A2 MULTI-FUNCTIONAL SMALL MOLECULES AS ANTI-PROLIFERATIVE AGENTS CURIS, INC. (US) 2008-03-20 WO disclosed
WO-2008033743-A1 SUBSTITUTED 2-INDOLINONE AS PTK INHIBITORS CONTAINING A ZINC BINDING MOIETY CURIS, INC. (US) 2008-03-20 WO disclosed