SCHEMBL8215550

SCHEMBL8215550

CCCc1ccc(NOCCc2ccc(N)cc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GFER P55789 1/20 0.42
CYP19A1 P11511 4/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
MAOB P27338 4/20 0.37
MAOA P21397 2/20 0.37
CA2 P00918 1/20 0.36
ALDH1A1 P00352 1/20 0.35
LPL P06858 1/20 0.34
LIPG Q9Y5X9 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27763969 0.79 TSHR (0.46) NPC1RAB9ACA2ALDH1A1MAPT
SCHEMBL27350060 0.78 GFER (0.52) GFERMAOBMAOACA2ALDH1A1
SCHEMBL5962 0.78 GFER (0.68) GFERCYP19A1MAOBMAOACA2
SCHEMBL16742377 0.76 MAPT (0.49) NPC1RAB9AALDH1A1MAPT
SCHEMBL29155827 0.75 GFER (0.65) GFERCYP19A1MAOBMAOACA2
SCHEMBL2026345 0.74 TDP1 (0.46) GFERCYP19A1NPC1RAB9AMAOA
SCHEMBL11935855 0.74 MAPT (0.49) GFERNPC1RAB9AMAOBMAOA
Ethylamine SCHEMBL27859952 0.73 GFER (0.62) GFERCYP19A1MAOBMAOACA2
SCHEMBL1979097 0.72 CYP3A4 (0.37) GFERRAB9AALDH1A1MAPT
SCHEMBL1696232 0.72 GFER (0.59) GFERCYP19A1NPC1RAB9AMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1019720-A1 COMBINATORIAL PROCESS FOR PREPARING TETRAHYDROQUINOLINE LIBRARIES ELI LILLY AND COMPANY (US) 2000-07-19 EP disclosed
WO-1998027427-A1 COMBINATORIAL PROCESS FOR PREPARING TETRAHYDROQUINOLINE LIBRARIES ELI LILLY AND COMPANY (US) 1998-06-25 WO disclosed