4-Hydroxyphenylmethylene Hydantoin

4-Hydroxyphenylmethylene Hydantoin

SCHEMBL8216459

O=C1NC(=O)/C(=C\c2ccc(O)cc2)N1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 9/20 1.00
METAP1 P53582 1/20 0.70
MAPT P10636 4/20 0.65
MEN1 O00255 3/20 0.65
KMT2A Q03164 3/20 0.65
BLM P54132 2/20 0.65
KDM4E B2RXH2 1/20 0.65
L3MBTL1 Q9Y468 1/20 0.65
CGAS Q8N884 1/20 0.62
LMNA P02545 3/20 0.62
RAB9A P51151 2/20 0.62
POLB P06746 1/20 0.62
CLK1 P49759 1/20 0.62
DYRK1A Q13627 1/20 0.62
SMN1; SMN2 Q16637 1/20 0.54
HPGD P15428 2/20 0.54
APAF1 O14727 1/20 0.54
ALDH1A1 P00352 1/20 0.54
THRB P10828 1/20 0.54
AKR1B1 P15121 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
4-Hydroxyphenylmethylene Hydantoin SCHEMBL5343815 1.00 GSK3B (1.00) GSK3BMETAP1MAPTMEN1KMT2A
4-Hydroxyphenylmethylene Hydantoin SCHEMBL5346095 1.00 GSK3B (1.00) GSK3BMETAP1MAPTMEN1KMT2A
SCHEMBL12821680 0.90 GSK3B (0.81) GSK3BMETAP1MAPTMEN1KMT2A
SCHEMBL12821679 0.90 GSK3B (0.81) GSK3BMETAP1MAPTMEN1KMT2A
SCHEMBL13848414 0.82 METAP1 (1.00) GSK3BMETAP1MAPTMEN1KMT2A
SCHEMBL15421390 0.81 GSK3B (0.69) GSK3BMETAP1MAPTMEN1KMT2A
SCHEMBL2873487 0.81 GSK3B (0.69) GSK3BMETAP1MAPTMEN1KMT2A
SCHEMBL15421387 0.81 GSK3B (0.69) GSK3BMETAP1MAPTMEN1KMT2A
SCHEMBL16685954 0.81 GSK3B (1.00) GSK3BMAPTMEN1KMT2ABLM
SCHEMBL8544557 0.81 GSK3B (1.00) GSK3BMAPTMEN1KMT2ABLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160102065-A1 NOVEL COMPOUND HAVING SKIN-WHITENING, ANTI-OXIDIZING AND PPAR ACTIVITIES AND MEDICAL USE THEREOF PUSAN NATIONAL UNIVERSITY INDUSTRY-UNIVERSITY COOPERATION FOUNDATION (KR) 2016-04-14 US claimed
US-8188130-B1 Anti-cancer hydantoin compounds and methods UNIVERSITY OF LOUISIANA AT MONROE (US) 2012-05-29 US claimed
US-9896421-B2 Compound having skin-whitening, anti-oxidizing and PPAR activities and medical use thereof PUSAN NATIONAL UNIVERSITY INDUSTRY-UNIVERSITY COOPERATION FOUNDATION (KR) 2018-02-20 US disclosed
US-20160102065-A1 NOVEL COMPOUND HAVING SKIN-WHITENING, ANTI-OXIDIZING AND PPAR ACTIVITIES AND MEDICAL USE THEREOF PUSAN NATIONAL UNIVERSITY INDUSTRY-UNIVERSITY COOPERATION FOUNDATION (KR) 2016-04-14 US disclosed
US-9216148-B2 Compound having skin-whitening, anti-oxidizing and PPAR activities and medical use therefor PUSAN NATIONAL UNIVERSITY INDUSTRY-UNIVERSITY COOPERATION FOUNDATION (KR) 2015-12-22 US disclosed
US-20140023603-A1 NOVEL COMPOUND HAVING SKIN-WHITENING, ANTI-OXIDIZING AND PPAR ACTIVITIES AND MEDICAL USE THEREFOR PUSAN NATIONAL UNIVERSITY INDUSTRY-UNIVERSITY COOPERATION FOUNDATION (KR) 2014-01-23 US disclosed
US-8188130-B1 Anti-cancer hydantoin compounds and methods UNIVERSITY OF LOUISIANA AT MONROE (US) 2012-05-29 US disclosed
US-8188130-B1 Anti-cancer hydantoin compounds and methods UNIVERSITY OF LOUISIANA AT MONROE (US) 2012-05-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140023603-A1 NOVEL COMPOUND HAVING SKIN-WHITENING, ANTI-OXIDIZING AND PPAR ACTIVITIES AND MEDICAL USE THEREFOR PPARG, PPARA, PPARD GSK3B 2733/4885METAP1 882/4885MAPT 2700/4885
US-20160102065-A1 NOVEL COMPOUND HAVING SKIN-WHITENING, ANTI-OXIDIZING AND PPAR ACTIVITIES AND MEDICAL USE THEREOF PPARG, PPARA, TYR GSK3B 3223/4885METAP1 983/4885MAPT 1956/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.