SCHEMBL8216655

SCHEMBL8216655

CC(O)(C(=O)NCC(F)(F)C(F)(F)F)C(=O)NC1CN(C(=O)OCC(F)(F)F)c2ccccc2N(CC(F)(F)F)C1=O

nearest known ligand 0.39

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 11/20 0.39
XIAP P98170 9/20 0.36
CYP3A4 P08684 4/20 0.36
SCN10A Q9Y5Y9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14093717 1.00 SCN9A (0.39) SCN9AXIAPCYP3A4SCN10A
SCHEMBL14093728 0.93 PSEN1 (0.40) SCN9AXIAPCYP3A4SCN10A
SCHEMBL14093721 0.92 XIAP (0.36) SCN9AXIAPCYP3A4
SCHEMBL8214145 0.92 XIAP (0.36) SCN9AXIAPCYP3A4
SCHEMBL8212213 0.89 SCN9A (0.33) SCN9AXIAP
SCHEMBL8209811 0.89 SCN9A (0.41) SCN9AXIAPCYP3A4SCN10A
SCHEMBL8207421 0.87 XIAP (0.38) SCN9AXIAPCYP3A4SCN10A
SCHEMBL8208458 0.85 XIAP (0.36) XIAPCYP3A4
SCHEMBL14093725 0.84 XIAP (0.35) XIAPCYP3A4
SCHEMBL8207647 0.84 XIAP (0.35) XIAPCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008034735-A2 4-OXO-2,3,4,5-TETRAHYDRO-BENZO[B][1,4]DIAZEPINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-03-27 WO disclosed