SCHEMBL8216972

SCHEMBL8216972

CCCCOCn1ncc(-c2nnc(O[C@H](C)c3cc(-c4cccc(C)c4)on3)n2C)cc1=O

nearest known ligand 0.62

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 10/20 0.62
KCNH2 Q12809 2/20 0.34
HRH3 Q9Y5N1 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP19A1 P11511 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13201363 0.92 GRM5 (0.63) GRM5KCNH2KMT2A
SCHEMBL2963963 0.92 GRM5 (0.63) GRM5KCNH2KMT2A
SCHEMBL13201362 0.84 GRM5 (0.66) GRM5KCNH2
SCHEMBL2966417 0.84 GRM5 (0.66) GRM5KCNH2
SCHEMBL2959176 0.77 GRM5 (1.00) GRM5KCNH2KMT2A
SCHEMBL13201365 0.73 GRM5 (0.62) GRM5KCNH2
SCHEMBL2956435 0.73 GRM5 (0.62) GRM5KCNH2
SCHEMBL2959556 0.72 GRM5 (1.00) GRM5KCNH2
SCHEMBL2967887 0.72 GRM5 (1.00) GRM5KCNH2
SCHEMBL13201361 0.72 GRM5 (0.66) GRM5KCNH2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008041075-A1 MGLUR5 MODULATORS ASTRAZENECA AB (SE) 2008-04-10 WO disclosed