SCHEMBL8220294

SCHEMBL8220294

CC1=C(C(=O)C2CCC2)[C@@H](c2ccc(C)cc2)NC(=O)N1c1cccc(C(F)(F)F)c1

nearest known ligand 0.62

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ELANE P08246 18/20 0.62
CYP2C9 P11712 6/20 0.62
ADRB1 P08588 1/20 0.55
HTR1A P08908 1/20 0.55
HRH3 Q9Y5N1 1/20 0.55
CYP2C8 P10632 1/20 0.52
CYP2C19 P33261 1/20 0.52
POLB P06746 1/20 0.45
CYP3A4 P08684 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3482549 0.90 ELANE (0.78) ELANECYP2C9ADRB1HTR1AHRH3
SCHEMBL395327 0.90 ELANE (0.78) ELANECYP2C9ADRB1HTR1AHRH3
SCHEMBL394597 0.87 ELANE (0.77) ELANECYP2C9ADRB1HTR1AHRH3
SCHEMBL14899950 0.87 ELANE (0.67) ELANECYP2C9ADRB1HTR1AHRH3
SCHEMBL393057 0.86 ELANE (0.81) ELANECYP2C9ADRB1HTR1AHRH3
SCHEMBL393056 0.86 ELANE (0.81) ELANECYP2C9ADRB1HTR1AHRH3
SCHEMBL395516 0.81 ELANE (0.72) ELANECYP2C9ADRB1HTR1AHRH3
SCHEMBL8056317 0.79 ELANE (0.65) ELANECYP2C9ADRB1HTR1AHRH3
SCHEMBL391892 0.78 ELANE (0.67) ELANECYP2C9ADRB1HTR1AHRH3
SCHEMBL4449580 0.77 ELANE (0.85) ELANECYP2C9ADRB1HTR1AHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008003412-A1 THE USE OF 1,4-DIARYL-DIHYDROPYRIMIDINE-2-ON DERIVATIVES FOR TREATING PULMONARY ARTERIAL HYPERTENSION BAYER HEALTHCARE AG (DE) 2008-01-10 WO disclosed