SCHEMBL8220767

SCHEMBL8220767

CNC(=O)N1CCCC2(CCNCC2)c2ccccc21

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 3/20 0.48
ROCK2 O75116 1/20 0.42
ROCK1 Q13464 1/20 0.42
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 1/20 0.39
AKT1 P31749 3/20 0.39
HSD11B1 P28845 1/20 0.39
CREBBP Q92793 3/20 0.38
CYP2D6 P10635 1/20 0.37
P2RY1 P47900 1/20 0.37
HDAC1 Q13547 2/20 0.36
HDAC8 Q9BY41 2/20 0.36
HDAC6 Q9UBN7 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2982201 0.86 NOTUM (0.62) NOTUMROCK2ROCK1AKT1HSD11B1
SCHEMBL6543320 0.86 NOTUM (0.57) NOTUMROCK2ROCK1AKT1P2RY1
SCHEMBL8225944 0.83 NOTUM (0.48) NOTUMROCK2ROCK1CYP1A2CYP3A4
SCHEMBL2984971 0.82 NOTUM (0.48) NOTUMROCK2ROCK1CYP1A2CYP3A4
SCHEMBL1713623 0.78 NOTUM (0.60) NOTUMROCK2ROCK1AKT1HSD11B1
SCHEMBL12316015 0.74 NOTUM (0.46) NOTUMROCK2ROCK1AKT1HSD11B1
SCHEMBL30232786 0.74 NOTUM (0.63) NOTUMROCK2ROCK1AKT1P2RY1
SCHEMBL1572534 0.74 NOTUM (0.63) NOTUMROCK2ROCK1AKT1P2RY1
SCHEMBL655024 0.73 NOTUM (0.80) NOTUMROCK2ROCK1AKT1P2RY1
SCHEMBL14529913 0.73 NOTUM (0.57) NOTUMROCK2ROCK1AKT1P2RY1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021545-A2 MODULATORS OF MUSCARINIC RECEPTORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-02-21 WO disclosed