SCHEMBL8229215

SCHEMBL8229215

Bc1ccc(F)cc1Cn1c(N2CCC[C@@H](N)C2)cc(=O)n(C)c1=O

nearest known ligand 0.79

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 20/20 0.79
DPP8 Q6V1X1 1/20 0.64
OPRM1 P35372 1/20 0.63
OPRK1 P41145 1/20 0.63
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
CYP2D6 P10635 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8228913 0.91 DPP4 (0.70) DPP4DPP8CYP1A2CYP3A4CYP2D6
SCHEMBL14142701 0.89 DPP4 (0.80) DPP4DPP8OPRM1OPRK1CYP1A2
SCHEMBL389715 0.88 DPP4 (1.00) DPP4DPP8OPRM1OPRK1CYP1A2
SCHEMBL2087382 0.88 DPP4 (1.00) DPP4DPP8OPRM1OPRK1CYP1A2
SCHEMBL389714 0.88 DPP4 (1.00) DPP4DPP8OPRM1OPRK1CYP1A2
SCHEMBL390403 0.88 DPP4 (1.00) DPP4DPP8OPRM1OPRK1CYP1A2
SCHEMBL8237899 0.87 DPP4 (0.78) DPP4DPP8OPRM1OPRK1
Trelagliptin SCHEMBL175726 0.87 DPP4 (1.00) DPP4DPP8OPRM1OPRK1CYP1A2
Trelagliptin SCHEMBL29349599 0.87 DPP4 (1.00) DPP4DPP8OPRM1OPRK1CYP1A2
Trelagliptin SCHEMBL175727 0.87 DPP4 (1.00) DPP4DPP8OPRM1OPRK1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007112368-A1 PREPARATION OF (R)-3-AMINOPIPERIDINE DIHYDROCHLORIDE TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-10-04 WO disclosed