SCHEMBL8229219

SCHEMBL8229219

CNc1c(C)cccc1N

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CD44 P16070 1/20 0.52
CYP3A4 P08684 5/20 0.48
TDP1 Q9NUW8 2/20 0.48
TSHR P16473 3/20 0.46
PIK3CA P42336 1/20 0.46
GRIN2D O15399 1/20 0.38
GRIN3B O60391 1/20 0.38
GRIN1 Q05586 1/20 0.38
GRIN2A Q12879 1/20 0.38
GRIN2B Q13224 1/20 0.38
GRIN2C Q14957 1/20 0.38
GRIN3A Q8TCU5 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
ALDH1A1 P00352 4/20 0.38
NPSR1 Q6W5P4 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP2A6 P11509 1/20 0.36
HPGD P15428 1/20 0.36
HSD17B10 Q99714 1/20 0.36
DPP4 P27487 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23030132 0.86 CD44 (0.52) CD44CYP3A4TDP1TSHRPIK3CA
SCHEMBL8466087 0.85 TSHR (0.48) CD44CYP3A4TDP1TSHRPIK3CA
SCHEMBL1006539 0.82 CYP1A2 (0.45) CD44CYP3A4TSHRGRIN2DGRIN3B
SCHEMBL8439291 0.81 CD44 (0.52) CD44CYP3A4TDP1TSHRPIK3CA
Benzene SCHEMBL28199279 0.79 CYP1A2 (0.43) CYP3A4TSHRGRIN2DGRIN3BGRIN1
SCHEMBL27839905 0.79 CYP1A2 (0.43) CD44CYP3A4TSHRGRIN2DGRIN3B
Hydrochloric Acid SCHEMBL2864880 0.79 CYP1A2 (0.43) CD44CYP3A4TDP1TSHRGRIN2D
SCHEMBL20120116 0.79 CD44 (0.50) CD44CYP3A4TDP1TSHRPIK3CA
SCHEMBL15089832 0.78 CYP3A4 (0.37) CD44CYP3A4TDP1TSHRPIK3CA
SCHEMBL11779941 0.76 CYP3A4 (0.40) CD44CYP3A4TDP1TSHRPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108779108-A 3- (2,3- dihydro -1H- indenes -5- bases) propanoic derivatives and their purposes as NRF2 conditioning agents 葛兰素史密斯克莱知识产权发展有限公司 2018-11-09 CN disclosed
CN-108137557-A Nrf2 modulators 葛兰素史密斯克莱知识产权发展有限公司 2018-06-08 CN disclosed
WO-2016134145-A9 ARTIFICIAL SELF-SUFFICIENT CYTOCHROME P450S UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2017-02-16 WO disclosed
CN-101155787-B (3,4-dihydro-quinazolin-2-yl)-indan-1-yl-amines HOFFMANN LA ROCHE 2010-11-24 CN disclosed
US-20090192169-A1 Bicyclic Benzimidazole Compounds and Their Use as Metabotropic Glutamate Receptor Potentiators ASTRAZENECA AB (SE) 2009-07-30 US disclosed
US-20090192169-A1 Bicyclic Benzimidazole Compounds and Their Use as Metabotropic Glutamate Receptor Potentiators ASTRAZENECA AB (SE) 2009-07-30 US disclosed
CN-101155787-A (3,4-dihydro-quinazolin-2-yl)-indan-1-yl-amines HOFFMANN LA ROCHE (CH) 2008-04-02 CN disclosed
WO-2007115077-A2 BICYCLIC BENZIMIDAZOLE COMPOUNDS AND THEIR USE AS METABOTROPIC GLUTAMATE RECEPTOR POTENTIATORS ASTRAZENECA AB (SE) 2007-10-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090192169-A1 Bicyclic Benzimidazole Compounds and Their Use as Metabotropic Glutamate Receptor Potentiators GRM1, GRIN1, GRM2 CD44 4455/4885CYP3A4 1310/4885TDP1 4163/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.