SCHEMBL8232123

SCHEMBL8232123

Cn1c(N2CCN(Cc3ccccc3)CC2)nc(-c2ccncc2F)cc1=O

nearest known ligand 0.54

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 18/20 0.54
CYP2D6 P10635 4/20 0.54
CYP1A2 P05177 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13711456 0.86 GSK3B (0.73) GSK3BCYP2D6CYP1A2
SCHEMBL13711452 0.86 GSK3B (0.70) GSK3BCYP2D6CYP1A2
SCHEMBL8228618 0.86 GSK3B (0.70) GSK3BCYP2D6CYP1A2
SCHEMBL1652648 0.83 GSK3B (0.58) GSK3BCYP2D6CYP1A2
SCHEMBL87782 0.82 GSK3B (0.54) GSK3BCYP2D6CYP1A2
SCHEMBL8268075 0.82 GSK3B (0.63) GSK3BCYP2D6CYP1A2
SCHEMBL87832 0.81 GSK3B (0.62) GSK3BCYP2D6CYP1A2
SCHEMBL81961 0.80 GSK3B (0.69) GSK3BCYP2D6CYP1A2
SCHEMBL699220 0.80 GSK3B (0.54) GSK3BCYP2D6CYP1A2
SCHEMBL698023 0.80 GSK3B (0.54) GSK3BCYP2D6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007119463-A1 2-(CYCLIC AMINO)-PYRIMIDONE DERIVATIVES AS TPK1 INHIBITORS MITSUBISHI TANABE PHARMA CORPORATION (JP) 2007-10-25 WO disclosed