SCHEMBL8234166

SCHEMBL8234166

COC(=O)C(Cc1ccc(CCCNc2ccccn2)cc1)NC(=O)c1c(Cl)cccc1Cl

nearest known ligand 0.77

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 19/20 0.77
ITGA5 P08648 16/20 0.77
ITGB3 P05106 4/20 0.69
ITGAV P06756 4/20 0.69
ITGB5 P18084 1/20 0.45
ITGB6 P18564 1/20 0.45
ITGA4 P13612 2/20 0.44
MDM4 O15151 1/20 0.44
MDM2 Q00987 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4068226 1.00 ITGB1 (0.77) ITGB1ITGA5ITGB3ITGAVITGB5
SCHEMBL8236797 0.97 ITGB1 (0.81) ITGB1ITGA5ITGB3ITGAVITGB5
SCHEMBL4067367 0.97 ITGB1 (0.81) ITGB1ITGA5ITGB3ITGAVITGB5
SCHEMBL14270716 0.91 ITGB1 (0.83) ITGB1ITGA5ITGB3ITGAVITGB5
SCHEMBL4066779 0.90 ITGB1 (0.94) ITGB1ITGA5ITGB3ITGAVITGA4
SCHEMBL8232202 0.90 ITGB1 (0.94) ITGB1ITGA5ITGB3ITGAVITGA4
SCHEMBL20025129 0.89 ITGB1 (0.70) ITGB1ITGA5ITGB3ITGAVITGB5
SCHEMBL8234167 0.89 ITGB1 (0.65) ITGB1ITGA5ITGB3ITGAVITGA4
SCHEMBL4068703 0.89 ITGB1 (0.65) ITGB1ITGA5ITGB3ITGAVITGA4
SCHEMBL8234588 0.89 ITGB1 (0.64) ITGB1ITGA5ITGB3ITGAVITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007141473-A1 N-(BENZOYL)-O- [2- (PYRIDIN- 2 -YLAMINO) ETHYL] -L-TYROSINE DERIVATIVES AND RELATED COMPOUNDS AS A5B1 ANTAGONISTS FOR THE TREATMENT OF SOLID TUMORS ASTRAZENECA AB (SE) 2007-12-13 WO disclosed